SCHEMBL27675111

SCHEMBL27675111

CC(C(=O)C(C)N1CCc2ccccc21)N1CCc2ccccc21

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.56
GFER P55789 1/20 0.56
NOTUM Q6P988 3/20 0.53
ALDH1A1 P00352 4/20 0.51
MAPT P10636 3/20 0.51
TSHR P16473 2/20 0.51
KDM4E B2RXH2 1/20 0.51
LMNA P02545 1/20 0.51
POLB P06746 2/20 0.51
L3MBTL1 Q9Y468 2/20 0.47
SMN1; SMN2 Q16637 4/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
TP53 P04637 2/20 0.46
NFKB1 P19838 2/20 0.46
NFKB2 Q00653 2/20 0.46
RELA Q04206 2/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 2/20 0.46
SLC6A2 P23975 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27643466 0.90 NOTUM (0.55) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL4143391 0.88 GAA (0.55) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL13802543 0.87 GAA (0.57) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL10165554 0.84 NOTUM (0.53) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL6262183 0.80 SLC6A2 (0.52) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL1102007 0.80 ALDH1A1 (0.48) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL10203776 0.79 NOTUM (0.58) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL4553227 0.79 NOTUM (0.54) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL28765957 0.78 ATAD2 (0.42) GAAGFERNOTUMALDH1A1MAPT
SCHEMBL27675235 0.78 ABHD6 (0.47) GAAGFERNOTUMTSHRLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 8 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-103641765-A Modulators of ATP-binding cassette transporters VERTEX PHARMA 2014-03-19 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-101421258-B Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYPSYS INC 2013-08-21 CN disclosed
CN-102652128-A 4-Oxo-1H-quinoline-3-carboxamides as modulators of ATP-binding cassette transporters VERTEX PHARMA 2012-08-29 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101421258-A Sulfonyl-substituted bicyclic compounds as PPAR modulators KALYSPSYS INC (US) 2009-04-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed