SCHEMBL27675213

SCHEMBL27675213

O=C(O)c1cn(C(=O)Nc2ccccc2-c2ccncc2)c2ccccc2c1=O

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.46
S1PR1 P21453 2/20 0.43
S1PR3 Q99500 2/20 0.43
CAPN1 P07384 1/20 0.41
LMNA P02545 1/20 0.41
ALDH1A1 P00352 3/20 0.40
ALOX15 P16050 1/20 0.40
TSHR P16473 1/20 0.40
KDM4E B2RXH2 3/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
ATM Q13315 1/20 0.39
CHRM1 P11229 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
FABP5 Q01469 1/20 0.38
HTR6 P50406 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27920808 0.87 KDM4E (0.41) S1PR1S1PR3LMNAALDH1A1KDM4E
SCHEMBL27693464 0.87 LMNA (0.44) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27675276 0.87 LMNA (0.42) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27693550 0.86 NTRK1 (0.43) S1PR1S1PR3LMNAALDH1A1
SCHEMBL27693577 0.86 LMNA (0.46) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27693531 0.85 CHRM1 (0.41) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27675140 0.84 ALDH1A1 (0.40) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27693536 0.84 KDM4E (0.39) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27675121 0.84 CHRM1 (0.47) S1PR1S1PR3CAPN1LMNAKDM4E
SCHEMBL27693494 0.84 LMNA (0.40) LMNAALDH1A1KDM4EPOLBHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed