SCHEMBL27675276

SCHEMBL27675276

O=C(O)c1cn(C(=O)Nc2ccccc2-c2ccc(F)cc2)c2ccccc2c1=O

nearest known ligand 0.50

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
LMNA P02545 3/20 0.42
ALDH1A1 P00352 2/20 0.42
TP53 P04637 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
NTRK1 P04629 1/20 0.40
KMT2A Q03164 1/20 0.40
KDM4E B2RXH2 3/20 0.39
POLB P06746 1/20 0.39
HPGD P15428 1/20 0.39
HSD17B10 Q99714 1/20 0.39
EP300 Q09472 1/20 0.38
CREBBP Q92793 1/20 0.38
CHRM1 P11229 1/20 0.38
FABP3 P05413 1/20 0.38
FABP4 P15090 1/20 0.38
FABP5 Q01469 1/20 0.38
HCAR2 Q8TDS4 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693464 0.89 LMNA (0.44) LMNAALDH1A1NPSR1KMT2AKDM4E
SCHEMBL27920808 0.89 KDM4E (0.41) LMNAALDH1A1TP53KMT2AKDM4E
SCHEMBL27693515 0.89 CREBBP (0.46) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27693550 0.89 NTRK1 (0.43) LMNAALDH1A1NTRK1CREBBP
SCHEMBL27693577 0.88 LMNA (0.46) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27693531 0.87 CHRM1 (0.41) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27675213 0.87 HTT (0.46) LMNAALDH1A1KDM4EPOLBHPGD
SCHEMBL27675161 0.87 POLB (0.43) LMNAALDH1A1KMT2AKDM4EPOLB
SCHEMBL27693536 0.86 KDM4E (0.39) LMNAALDH1A1KMT2AKDM4EPOLB
SCHEMBL27675140 0.86 ALDH1A1 (0.40) LMNAALDH1A1KMT2AKDM4EPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101891680-B Modulators of ATP-binding cassette transporters VERTEX PHARMACEUTICALS INCORPORATED (US) 2014-10-29 CN disclosed
CN-101935301-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2013-10-16 CN disclosed
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed