SCHEMBL27675331

SCHEMBL27675331

O=C(O)c1cn(C(=O)Nc2ccccc2-c2ccccc2OC(F)(F)F)c2ccccc2c1=O

nearest known ligand 0.41

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
CFD P00746 6/20 0.41
FABP4 P15090 1/20 0.41
FABP5 Q01469 1/20 0.41
CYP2C9 P11712 1/20 0.40
DHODH Q02127 1/20 0.39
LMNA P02545 1/20 0.38
RORC P51449 2/20 0.37
S1PR1 P21453 2/20 0.37
S1PR3 Q99500 2/20 0.37
SCN10A Q9Y5Y9 1/20 0.37
KDM4E B2RXH2 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
HPGD P15428 1/20 0.36
HSD17B10 Q99714 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27675229 0.87 KDM4E (0.45) LMNAKDM4EALDH1A1POLBHPGD
SCHEMBL27675221 0.86 SERPINE1 (0.42) CFDLMNAS1PR1S1PR3
SCHEMBL27693557 0.86 LMNA (0.40) LMNAKDM4EALDH1A1POLBHPGD
SCHEMBL28766939 0.85 S1PR1 (0.43) CYP2C9LMNAS1PR1S1PR3KDM4E
SCHEMBL28766933 0.84 CFD (0.42) CFDCYP2C9
SCHEMBL27675161 0.83 POLB (0.43) LMNAKDM4EALDH1A1POLBHPGD
SCHEMBL27675276 0.81 LMNA (0.42) FABP4FABP5LMNAKDM4EALDH1A1
SCHEMBL27991300 0.81 KDM4E (0.43) CYP2C9LMNAKDM4EALDH1A1POLB
SCHEMBL27693550 0.81 NTRK1 (0.43) CFDLMNAS1PR1S1PR3ALDH1A1
SCHEMBL27693793 0.80 KMT2A (0.51) LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed