SCHEMBL27675229

SCHEMBL27675229

COc1ccccc1-c1ccccc1NC(=O)n1cc(C(=O)O)c(=O)c2ccccc21

nearest known ligand 0.47

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 5/20 0.45
CHRM1 P11229 1/20 0.44
ALDH1A1 P00352 5/20 0.44
MCL1 Q07820 2/20 0.42
BAD Q92934 2/20 0.42
KMT2A Q03164 4/20 0.42
MEN1 O00255 2/20 0.42
CLCN2 P51788 1/20 0.41
CASP3 P42574 1/20 0.41
HPGD P15428 2/20 0.41
HSD17B10 Q99714 2/20 0.41
POLB P06746 1/20 0.41
LMNA P02545 1/20 0.40
CDC25B P30305 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
GPR35 Q9HC97 1/20 0.40
GAA P10253 1/20 0.40
CYP3A4 P08684 1/20 0.40
THRB P10828 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27693793 0.91 KMT2A (0.51) KDM4ECHRM1KMT2AMEN1CASP3
SCHEMBL27693557 0.88 LMNA (0.40) KDM4ECHRM1ALDH1A1HPGDHSD17B10
SCHEMBL27675331 0.87 CFD (0.41) KDM4EALDH1A1HPGDHSD17B10POLB
SCHEMBL27675114 0.86 CHRM1 (0.39) KDM4ECHRM1ALDH1A1KMT2AMEN1
SCHEMBL27991300 0.86 KDM4E (0.43) KDM4ECHRM1ALDH1A1MCL1BAD
SCHEMBL27675161 0.84 POLB (0.43) KDM4ECHRM1ALDH1A1KMT2AMEN1
SCHEMBL27693506 0.83 CREBBP (0.49) KDM4ECHRM1ALDH1A1MCL1BAD
SCHEMBL27920808 0.82 KDM4E (0.41) KDM4EALDH1A1MCL1BADKMT2A
SCHEMBL27675276 0.82 LMNA (0.42) KDM4ECHRM1ALDH1A1KMT2AHPGD
SCHEMBL27693782 0.81 L3MBTL1 (0.44) KDM4ECHRM1ALDH1A1KMT2AMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101006076-B Modulators of ATP-binding cassette transporters VERTEX PHARMA 2010-09-29 CN disclosed
CN-101006076-A Modulators of ATP-binding cassette transporters VERTEX PHARMA (US) 2007-07-25 CN disclosed