SCHEMBL27684142

SCHEMBL27684142

COc1ccc(-c2cccc(C=CC#N)c2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ABL1 P00519 1/20 0.50
ABCB1 P08183 1/20 0.50
BCR P11274 1/20 0.50
ENPP2 Q13822 1/20 0.49
RELA Q04206 4/20 0.49
NFE2L2 Q16236 2/20 0.45
APP P05067 1/20 0.45
FDPS P14324 1/20 0.44
HDAC4 P56524 1/20 0.44
HDAC2 Q92769 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
TRPA1 O75762 1/20 0.42
PGR P06401 1/20 0.41
AR P10275 1/20 0.41
ERCC5 P28715 1/20 0.41
FEN1 P39748 1/20 0.41
NPC1 O15118 1/20 0.41
RAB9A P51151 1/20 0.41
MAOB P27338 1/20 0.40
CYP1A1 P04798 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27684133 0.84 FDPS (0.57) ABCB1ENPP2RELANFE2L2APP
SCHEMBL8928081 0.82 RELA (0.61) ENPP2RELANFE2L2FDPSCYP1A1
SCHEMBL8928082 0.82 RELA (0.61) ENPP2RELANFE2L2FDPSCYP1A1
SCHEMBL8904307 0.82 ENPP2 (0.54) ENPP2NFE2L2FDPSHDAC4HDAC2
SCHEMBL8904305 0.82 ENPP2 (0.54) ENPP2NFE2L2FDPSHDAC4HDAC2
SCHEMBL27698353 0.80 ENPP2 (0.49) ENPP2FDPSHDAC2HDAC8MAOB
SCHEMBL27745334 0.79 ENPP2 (0.40) ENPP2FDPSNPC1RAB9AMAOB
SCHEMBL442274 0.78 KDM4E (0.57) ABL1ABCB1BCRRELANFE2L2
SCHEMBL442275 0.78 KDM4E (0.57) ABL1ABCB1BCRRELANFE2L2
SCHEMBL694393 0.78 ENPP2 (0.50) ENPP2RELANFE2L2FDPSHDAC2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101053558-A Diphenylethylene compounds and uses thereof CELGENE CORP (US) 2007-10-17 CN disclosed