SCHEMBL2769178

SCHEMBL2769178

COC(=O)CCc1ccccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMN1; SMN2 Q16637 3/20 0.52
ALDH1A1 P00352 3/20 0.52
HRH3 Q9Y5N1 1/20 0.51
CYP1A2 P05177 3/20 0.51
LMNA P02545 2/20 0.51
TDP1 Q9NUW8 2/20 0.51
CYP2C19 P33261 1/20 0.51
ALOX15 P16050 2/20 0.50
TAAR1 Q96RJ0 1/20 0.50
TSHR P16473 1/20 0.49
POLB P06746 1/20 0.48
MEN1 O00255 1/20 0.48
KMT2A Q03164 1/20 0.48
HPGD P15428 1/20 0.48
KDM4E B2RXH2 1/20 0.48
HRH1 P35367 1/20 0.47
NPC1 O15118 2/20 0.47
RAB9A P51151 2/20 0.47
MAPK1 P28482 1/20 0.47
HTT P42858 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL2769175 0.98 ALDH1A1 (0.53) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL18163286 0.90 SMN1; SMN2 (0.60) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL6643882 0.87 SMN1; SMN2 (0.55) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL22578221 0.86 CYP1A2 (0.54) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL11769016 0.86 CYP1A2 (0.54) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL11532136 0.84 TDP1 (0.55) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL4341122 0.83 LMNA (0.57) SMN1; SMN2ALDH1A1CYP1A2LMNATDP1
SCHEMBL14640301 0.83 HRH1 (0.52) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL9411265 0.83 CYP1A2 (0.51) SMN1; SMN2ALDH1A1HRH3CYP1A2LMNA
SCHEMBL78000 0.82 SMN1; SMN2 (0.53) SMN1; SMN2ALDH1A1CYP1A2LMNACYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 36 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-5939268-A DIELS-ALDER REACTION PRODUCT OF A DIENE AND A DIENOPHILE; CHEMICAL INTERMEDIATES FOR DRUGS, SOLID PHASE SYNTHESIS THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US claimed
EP-0773953-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS INSTITUTE (US) 1997-05-21 EP claimed
WO-1996003424-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS RESEARCH INSTITUTE (US) 1996-02-08 WO claimed
CN-116685576-A Cysteine protease inhibitors and methods of use thereof 美商帕迪斯生物科学公司 2023-09-01 CN disclosed
CN-107709334-B Novel amino acid derivatives, process for their preparation and pharmaceutical compositions containing them 法国施维雅药厂 2021-04-13 CN disclosed
US-9957217-B2 Conversion of alcohols to carboxylic acids using heterogeneous palladium-based catalysts WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2018-05-01 US disclosed
WO-2017214359-A1 NOVEL CLOSTRIDIUM DIFFICILE TOXIN INHIBITORS VENENUM BIODESIGN LLC (US) 2017-12-14 WO disclosed
US-20170137362-A1 CONVERSION OF ALCOHOLS TO CARBOXYLIC ACIDS USING HETEROGENEOUS PALLADIUM-BASED CATALYSTS WISCONSIN ALUMNI RESEARCH FOUNDATION 2017-05-18 US disclosed
US-9593064-B2 Conversion of alcohols to alkyl esters and carboxylic acids using heterogeneous palladium-based catalysts WISCONSIN ALUMNI RESEARCH FOUNDATION (US) 2017-03-14 US disclosed
EP-2776389-B1 ARYL UREA DERIVATIVES AS N-FORMYL PEPTIDE RECEPTOR LIKE-1 (FPRL-1) RECEPTOR MODULATORS ALLERGAN INC (US) 2016-09-21 EP disclosed
US-20150314272-A1 Conversion Of Alcohols To Alkyl Esters And Carboxylic Acids Using Heterogeneous Palladium-Based Catalysts WISCONSIN ALUMNI RESEARCH FOUNDATION 2015-11-05 US disclosed
WO-2004012663-A2 HYDANTOIN DERIVATIVES AS INHIBITORS OF MATRIX METALLOPROTEINASES AND/OR TNF-ALPHA CONVERTING ENZYME BRISTOL-MYERS SQUIBB COMPANY (US) 2004-02-12 WO disclosed
US-5939268-A DIELS-ALDER REACTION PRODUCT OF A DIENE AND A DIENOPHILE; CHEMICAL INTERMEDIATES FOR DRUGS, SOLID PHASE SYNTHESIS THE SCRIPPS RESEARCH INSTITUTE (US) 1999-08-17 US disclosed
EP-0773953-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS INSTITUTE (US) 1997-05-21 EP disclosed
US-5624922-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1997-04-29 US disclosed
EP-0597540-B1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC (US) 1996-06-05 EP disclosed
WO-1996003424-A1 COMBINATORIAL LIBRARIES OF MOLECULES AND METHODS FOR PRODUCING SAME THE SCRIPPS RESEARCH INSTITUTE (US) 1996-02-08 WO disclosed
US-5380721-A Aryl-fused and hetaryl-fused-2,4-diazepine and 2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1995-01-10 US disclosed
EP-0597540-A1 Aryl-fused and hetaryl-fused-2,4-diazocine antiarrhythmic agents STERLING WINTHROP INC. (US) 1994-05-18 EP disclosed
US-4153795-A Cobalt pyridyl catalysts for hydroformylation DIRECTOR-GENERAL OF THE AGENCY OF INDUSTRIAL SCIENCE AND TECHNOLOGY (JP) 1979-05-08 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150314272-A1 Conversion Of Alcohols To Alkyl Esters And Carboxylic Acids Using Heterogeneous Palladium-Based Catalysts ADH5, ADH1A, ADH1C SMN1; SMN2 3152/4885ALDH1A1 391/4885HRH3 84/4885
US-20170137362-A1 CONVERSION OF ALCOHOLS TO CARBOXYLIC ACIDS USING HETEROGENEOUS PALLADIUM-BASED CATALYSTS ADH5, ADH1A, ADH1C SMN1; SMN2 3295/4885ALDH1A1 296/4885HRH3 88/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.