Piperidine

Piperidine

SCHEMBL2772399

C1CCNCC1.C=CC(N)=O.C=CC(N)=O

nearest known ligand 0.55

Full drug profile on Sugi Atlas →

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.55
TSHR P16473 1/20 0.55
FGFR4 P22455 1/20 0.55
KDM4E B2RXH2 2/20 0.35
KMT2A Q03164 2/20 0.35
MAPT P10636 1/20 0.35
ATM Q13315 1/20 0.35
CYP2D6 P10635 1/20 0.35
CA2 P00918 1/20 0.33
CHKA P35790 1/20 0.33
CXCR4 P61073 1/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
LMNA P02545 1/20 0.30
EPHX1 P07099 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Piperidine SCHEMBL8573009 1.00 ALDH1A1 (0.55) ALDH1A1TSHRFGFR4KDM4EKMT2A
Pyrrolidine SCHEMBL28160131 0.97 ALDH1A1 (0.58) ALDH1A1TSHRFGFR4KDM4EKMT2A
Acrylamide SCHEMBL25213622 0.92
Acrylamide SCHEMBL12544993 0.89
Piperazine SCHEMBL905449 0.87 ALDH1A1 (0.65) ALDH1A1TSHRFGFR4KDM4EKMT2A
Piperazine SCHEMBL8010364 0.87 ALDH1A1 (0.65) ALDH1A1TSHRFGFR4KDM4EKMT2A
Cyclohexane SCHEMBL2246750 0.84 ALDH1A1 (0.79) ALDH1A1TSHRFGFR4LMNAEPHX1
Cyclohexane SCHEMBL346356 0.84 ALDH1A1 (0.79) ALDH1A1TSHRFGFR4LMNAEPHX1
Piperidine SCHEMBL4407343 0.82 LMNA (0.53) ALDH1A1TSHRFGFR4KMT2AMAPT
Piperidine SCHEMBL3283269 0.81 ALDH1A1 (0.60) ALDH1A1TSHRKDM4EKMT2AMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 23 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120321533-A1 CATALYST ALMQVIST FREDRIK (SE) 2012-12-20 US claimed
JP-2010526659-A 2010-08-05 JP claimed
US-20100119424-A1 CATALYST ALMQUEST AB (SE) 2010-05-13 US claimed
EP-2152410-A2 PROCESS FOR THE PRODUCTION OF PALLADIUM SUPPORTED CATALYSTS FOR CATALYZING HECK, SUZUKI-MIYAURA SONOGASHIRA COUPLING AND BUCHWALD-HARTWIG REACTIONS Nordic chemquest Aktiebolag (SE) 2010-02-17 EP claimed
EP-1994983-A1 Catalyst containing covalently bonded formate groups and Pd(0) and process for its obtention Almquest AB (SE) 2008-11-26 EP claimed
WO-2008138938-A2 PROCESS FOR THE PRODUCTION OF PALLADIUM SUPPORTED CATALYSTS FOR CATALYZING HECK, SUZUKI-MIYAURA SONOGASHIRA COUPLING AND BUCHWALD-HARTWIG REACTIONS NORDIC CHEMQUEST AB (SE) 2008-11-20 WO claimed
EP-2682458-B1 CELL SHEET HAVING HYALURONIC ACID PRODUCTION ABILITY AND METHOD FOR PREPARING THE SAME CELLSEED INC (JP) 2019-10-23 EP disclosed
US-20140056858-A1 CELL SHEET HAVING HYALURONIC ACID PRODUCTION ABILITY AND METHOD FOR PREPARING THE SAME NATIONAL UNIVERSITY CORPORATION HOKKAIDO UNIVERSITY (JP) 2014-02-27 US disclosed
US-20130309703-A1 NOVEL METHOD FOR ANALYZING GLYCOSAMINOGLYCAN CELLSEED, INC. (JP) 2013-11-21 US disclosed
EP-2642286-A1 NOVEL METHOD FOR ANALYZING GLYCOSAMINOGLYCAN CellSeed Inc. (JP) 2013-09-25 EP disclosed
US-20120321533-A1 CATALYST ALMQVIST FREDRIK (SE) 2012-12-20 US disclosed
US-20100320373-A1 MASS SPECTROMETRIC QUANTITATIVE DETECTION OF METHYL MALONIC ACID AND SUCCINIC ACID USING HILIC ON A ZWITTERIONIC STATIONARY PHASE MERCK PATENT GESELLSCHAFT (DE) 2010-12-23 US disclosed
US-20100300971-A1 Zwitterionic stationary phase as well as method for using and producing said phase SEQUANT AB (SE) 2010-12-02 US disclosed
WO-2008138938-A2 PROCESS FOR THE PRODUCTION OF PALLADIUM SUPPORTED CATALYSTS FOR CATALYZING HECK, SUZUKI-MIYAURA SONOGASHIRA COUPLING AND BUCHWALD-HARTWIG REACTIONS NORDIC CHEMQUEST AB (SE) 2008-11-20 WO disclosed
WO-2008101736-A1 MASS SPECTROMETRIC QUANTITATIVE DETECTION OF METHYL MALONIC ACID AND SUCCINIC ACID USING HILIC ON A ZWITTERIONIC STATIONARY PHASE MERCK PATENT GMBH (DE) 2008-08-28 WO disclosed
EP-1962097-A1 Mass spectrometric quantitative detection of methyl malonic acid and succinic acid using hilic on a zwitterionic stationary phase SeQuant AB (SE) 2008-08-27 EP disclosed
EP-1137466-B1 A CHROMATOGRAPHY METHOD AND A COLUMN MATERIAL USEFUL IN SAID METHOD SEQUANT AB (SE) 2006-08-23 EP disclosed
US-6884345-B1 Chromatography method and a column material useful in said method MERCK PATENT GMBH (DE) 2005-04-26 US disclosed
EP-1137466-A1 A CHROMATOGRAPHY METHOD AND A COLUMN MATERIAL USEFUL IN SAID METHOD Irgum, Knut (SE) 2001-10-04 EP disclosed
WO-2000027496-A1 A CHROMATOGRAPHY METHOD AND A COLUMN MATERIAL USEFUL IN SAID METHOD IRGUM KNUT (SE) 2000-05-18 WO disclosed