SCHEMBL2773025

SCHEMBL2773025

Cc1cc(C(=O)O)ccc1-c1cscc1C.Cc1ccccc1-c1ccc(C(=O)O)cc1[N+](=O)[O-]

nearest known ligand 0.52

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
TSHR P16473 2/20 0.52
MEN1 O00255 3/20 0.46
KMT2A Q03164 3/20 0.46
POLB P06746 3/20 0.46
CASP6 P55212 2/20 0.46
CES2 O00748 1/20 0.45
CES1 P23141 1/20 0.45
HCAR3 P49019 7/20 0.43
LMNA P02545 1/20 0.43
TLR9 Q9NR96 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
ALDH1A1 P00352 3/20 0.42
EIF4E P06730 1/20 0.42
MAPT P10636 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2772166 0.89 TSHR (0.65) TSHRMEN1KMT2APOLBCASP6
SCHEMBL2771400 0.81 ESR1 (0.50) TSHRMEN1KMT2AL3MBTL1ALDH1A1
SCHEMBL5696841 0.79 TSHR (0.65) TSHRMEN1KMT2APOLBCASP6
SCHEMBL272092 0.78 TTR (0.56) TSHRKMT2APOLBCES2CES1
SCHEMBL6555682 0.77 POLB (0.59) TSHRPOLBCASP6HCAR3LMNA
SCHEMBL6555690 0.77 POLB (0.59) TSHRPOLBCASP6HCAR3LMNA
Hydrochloric Acid SCHEMBL9784149 0.77 CASP6 (0.62) TSHRPOLBCASP6HCAR3LMNA
SCHEMBL11195885 0.76 CASP6 (0.75) TSHRCASP6HCAR3LMNA
SCHEMBL2773008 0.75 VCAM1 (0.54) MEN1KMT2APOLBCES2CES1
SCHEMBL99918 0.72 CASP6 (0.64) TSHRPOLBCASP6HCAR3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2193125-A2 OXADIAZOLE DERIVATIVES Merck Serono S.A. (CH) 2010-06-09 EP disclosed
WO-2009043889-A2 OXADIAZOLE DERIVATIVES MERCK SERONO S.A. (CH) 2009-04-09 WO disclosed