SCHEMBL27751998

SCHEMBL27751998

CCc1[c]c(CN)cc(C(F)(F)F)c1

nearest known ligand 0.33

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.33
GABRB3 P28472 2/20 0.33
GABRA2 P47869 1/20 0.33
GABRB2 P47870 1/20 0.33
PTPN5 P54829 1/20 0.32
TAAR1 Q96RJ0 2/20 0.31
RAPGEF4 Q8WZA2 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL509184 0.90 GABRB3 (0.37) IDO1GABRB3GABRA2GABRB2PTPN5
SCHEMBL27751982 0.81
SCHEMBL4195232 0.78 RAPGEF4 (0.34) IDO1GABRB3GABRA2GABRB2PTPN5
SCHEMBL27731409 0.78 LOXL2 (0.30)
SCHEMBL28090050 0.75 TAAR1 (0.33) TAAR1
SCHEMBL27741441 0.75 TAAR1 (0.36) TAAR1
SCHEMBL289403 0.74
SCHEMBL27752027 0.74 PNMT (0.30)
SCHEMBL28776141 0.72 LOX (0.34)
SCHEMBL27731414 0.72 CA2 (0.41)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101448818-A New heterocyclic compounds for the inhibition of integrins and use thereof JERINI AG (DE) 2009-06-03 CN claimed
CN-101379056-A Compounds for the inhibition of integrins and use thereof JERINI AG (DE) 2009-03-04 CN claimed
CN-101448818-A New heterocyclic compounds for the inhibition of integrins and use thereof JERINI AG (DE) 2009-06-03 CN disclosed
CN-101379056-A Compounds for the inhibition of integrins and use thereof JERINI AG (DE) 2009-03-04 CN disclosed