SCHEMBL2776308

SCHEMBL2776308

CC(=O)C(C)(C)Nc1c(C(C)C)cccc1C(C)C

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 2/20 0.49
KMT2A Q03164 2/20 0.49
SMN1; SMN2 Q16637 1/20 0.49
GABRA1 P14867 2/20 0.42
GABRB2 P47870 2/20 0.42
FAAH O00519 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
HPGD P15428 1/20 0.42
TSHR P16473 1/20 0.42
GABRB1 P18505 1/20 0.42
GABRG2 P18507 1/20 0.42
PTGS1 P23219 1/20 0.42
SLC6A2 P23975 1/20 0.42
HTR2C P28335 1/20 0.42
GABRB3 P28472 1/20 0.42
GABRA5 P31644 1/20 0.42
GABRA3 P34903 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2243681 0.78 LMNA (0.40) LMNAKMT2ASMN1; SMN2GABRA1GABRB2
SCHEMBL2243684 0.78 LMNA (0.40) LMNAKMT2ASMN1; SMN2GABRA1GABRB2
SCHEMBL2243687 0.78 LMNA (0.40) LMNAKMT2ASMN1; SMN2GABRA1GABRB2
SCHEMBL1726368 0.75 KMT2A (0.62) LMNAKMT2ASMN1; SMN2MEN1TDP1
SCHEMBL21158254 0.75 GABRA1 (0.41) LMNAKMT2ASMN1; SMN2GABRA1GABRB2
SCHEMBL901604 0.74 KMT2A (0.57) LMNAKMT2ASMN1; SMN2MEN1TDP1
SCHEMBL14525630 0.73 SOAT2 (0.40) LMNAKMT2ASMN1; SMN2GABRA1GABRB2
SCHEMBL462304 0.72 LPAR1 (0.66) LMNAKMT2ASMN1; SMN2MEN1TDP1
SCHEMBL6429941 0.72 KMT2A (0.65) LMNAKMT2ASMN1; SMN2MEN1TDP1
SCHEMBL8845511 0.71 KMT2A (0.68) LMNAKMT2ASMN1; SMN2MEN1TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2170604-B1 ETHYLENE/ALPHA-OLEFIN INTERPOLYMERS HAVING LOW CRYSTALLINITY HARD BLOCKS DOW GLOBAL TECHNOLOGIES LLC (US) 2019-05-15 EP disclosed
EP-2179013-B1 LUBRICANT COMPOSITIONS DOW GLOBAL TECHNOLOGIES LLC (US) 2016-04-13 EP disclosed
US-8486878-B2 Viscosity index improver for lubricant compositions DOW GLOBAL TECHNOLOGIES, LLC (US) 2013-07-16 US disclosed
US-8476393-B2 Ethylene/α-olefin interpolymers containing low crystallinity hard blocks DOW GLOBAL TECHNOLOGIES, LLC (US) 2013-07-02 US disclosed
US-20100197540-A1 VISCOSITY INDEX IMPROVER FOR LUBRICANT COMPOSITIONS DOW GLOBAL TECHNOLOGIES LLC 2010-08-05 US disclosed
US-20100197880-A1 ETHYLENE/a- OLEFIN INTERPOLYMERS CONTAINING LOW CRYSTALI.INITY HARD BLOCKS DOW GLOBAL TECHNOLOGIES LLC 2010-08-05 US disclosed
EP-2179013-A1 VISCOSITY INDEX IMPROVER FOR LUBRICANT COMPOSITIONS Dow Global Technologies Inc. (US) 2010-04-28 EP disclosed
EP-2170604-A1 ETHYLENE/A-OLEFIN INTERPOLYMERS CONTAINING LOW CRYSTALLINITY HARD BLOCKS Dow Global Technologies Inc. (US) 2010-04-07 EP disclosed
WO-2009012215-A1 ETHYLENE/A-OLEFIN INTERPOLYMERS CONTAINING LOW CRYSTALLINITY HARD BLOCKS DOW GLOBAL TECHNOLOGIES INC. (US) 2009-01-22 WO disclosed
WO-2009012216-A1 VISCOSITY INDEX IMPROVER FOR LUBRICANT COMPOSITIONS DOW GLOBAL TECHNOLOGIES INC. (US) 2009-01-22 WO disclosed
US-7199255-B2 Imino-amide catalysts for olefin polymerization UNIVATION TECHNOLOGIES, LLC (US) 2007-04-03 US disclosed
US-7199255-B2 Imino-amide catalysts for olefin polymerization UNIVATION TECHNOLOGIES, LLC (US) 2007-04-03 US disclosed