SCHEMBL27768669

SCHEMBL27768669

COC(=O)Cc1c(C)n(C(=O)c2ccc(C)cc2)c2ccc(O)cc12

nearest known ligand 0.78

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 6/20 0.78
AKR1C2 P52895 3/20 0.78
PTGS2 P35354 11/20 0.65
CNR2 P34972 1/20 0.65
PTGS1 P23219 3/20 0.64
MAPT P10636 1/20 0.55
LMNA P02545 1/20 0.52
CYP1A2 P05177 1/20 0.52
CYP2D6 P10635 1/20 0.52
CYP2C9 P11712 1/20 0.52
TSHR P16473 1/20 0.52
NFKB1 P19838 1/20 0.52
HIF1A Q16665 1/20 0.52
NPSR1 Q6W5P4 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13448804 0.92 AKR1C3 (0.83) AKR1C3AKR1C2PTGS2CNR2MAPT
SCHEMBL20259423 0.91 PTGS2 (0.78) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL16656482 0.87 AKR1C3 (1.00) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL15062608 0.87 AKR1C3 (0.69) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL4055730 0.87 PTGS1 (0.82) AKR1C3AKR1C2PTGS2PTGS1MAPT
SCHEMBL25873193 0.85 PTGS2 (0.80) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL13195816 0.80 PTGS2 (0.74) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL17369559 0.79 PTGS2 (0.73) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL30761037 0.79 AKR1C3 (0.87) AKR1C3AKR1C2PTGS2CNR2PTGS1
SCHEMBL30426824 0.79 PTGS2 (1.00) AKR1C3AKR1C2PTGS2CNR2PTGS1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102850324-A Indole compounds MICROBIA INC 2013-01-02 CN disclosed
CN-101563337-A Indole compounds MICROBIA INC (US) 2009-10-21 CN disclosed