SCHEMBL27773232

SCHEMBL27773232

CC(C)(C)OC(=O)N1CCN(c2ccc3c(c2)CCN3C(=O)O)C(Cc2ccccc2)C1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ABHD6 Q9BV23 1/20 0.43
DAGLA Q9Y4D2 1/20 0.43
NR1H2 P55055 2/20 0.42
NR1H3 Q13133 2/20 0.42
GPR119 Q8TDV5 8/20 0.41
PARP1 P09874 1/20 0.39
JAK2 O60674 1/20 0.39
JAK1 P23458 1/20 0.39
DHODH Q02127 1/20 0.38
SMARCA2 P51531 1/20 0.38
SMARCA4 P51532 1/20 0.38
PBRM1 Q86U86 1/20 0.38
USP30 Q70CQ3 3/20 0.38
RORC P51449 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2949575 0.95 ABHD6 (0.44) ABHD6DAGLANR1H2NR1H3GPR119
SCHEMBL2946591 0.78 SLC6A4 (0.56) ABHD6DAGLANR1H2NR1H3PARP1
SCHEMBL31330650 0.77 ALDH1A1 (0.51) GPR119RORC
SCHEMBL2946903 0.75 SLC6A4 (0.46) ABHD6DAGLANR1H2NR1H3GPR119
SCHEMBL2948211 0.75 SLC6A2 (0.42) ABHD6DAGLANR1H2NR1H3PARP1
SCHEMBL31330699 0.74 NPC1 (0.56) GPR119
SCHEMBL23854712 0.73 TMEM97 (0.56) PARP1
SCHEMBL21800237 0.73 TMEM97 (0.56) PARP1
SCHEMBL21591745 0.72 HDAC1 (0.44) NR1H2GPR119USP30RORC
SCHEMBL8236259 0.72 GPR119 (0.52) NR1H2GPR119JAK2JAK1SMARCA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101501008-B Arylpiperazine derivatives and uses thereof F. HOFFMANN-LA ROCHE AG (CH) 2011-12-07 CN disclosed
CN-101501008-A Arylpiperazine derivatives and uses thereof HOFFMANN LA ROCHE (CH) 2009-08-05 CN disclosed