SCHEMBL27776366

SCHEMBL27776366

CC(CC(C)(C)OC(N)=O)c1ccccc1Br

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTT P42858 2/20 0.40
CYP2C19 P33261 2/20 0.39
CYP2C9 P11712 1/20 0.39
ALDH1A1 P00352 2/20 0.35
CYP3A4 P08684 1/20 0.35
ALOX15 P16050 1/20 0.35
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
AAK1 Q2M2I8 1/20 0.33
IDO1 P14902 1/20 0.33
TDO2 P48775 1/20 0.33
CYP26A1 O43174 2/20 0.32
POLB P06746 1/20 0.32
MEN1 O00255 1/20 0.32
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
KMT2A Q03164 1/20 0.32
CA12 O43570 1/20 0.32
CA1 P00915 1/20 0.32
CA2 P00918 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30998996 0.88 HTT (0.33) HTTCYP2C19CYP2C9
SCHEMBL27796919 0.81 APLNR (0.37) CYP2C19CYP3A4AAK1KMT2A
SCHEMBL27666222 0.79 RIPK1 (0.46) ALDH1A1CYP1A2CYP2D6POLB
SCHEMBL27666213 0.79 RIPK1 (0.46) ALDH1A1CYP1A2CYP2D6POLB
SCHEMBL25222546 0.77 ALOX5 (0.43) CYP2C19CYP2C9ALDH1A1CYP1A2CYP2D6
SCHEMBL27828808 0.77 ALOX5 (0.43) CYP2C19CYP2C9ALDH1A1CYP1A2CYP2D6
SCHEMBL25222547 0.77 ALOX5 (0.43) CYP2C19CYP2C9ALDH1A1CYP1A2CYP2D6
SCHEMBL3651052 0.76 CYP1A2 (0.47) HTTCYP2C19CYP2C9ALDH1A1CYP3A4
SCHEMBL27931107 0.76 APLNR (0.43) HTTALDH1A1AAK1MEN1NPC1
SCHEMBL27931106 0.76 APLNR (0.43) HTTALDH1A1AAK1MEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101679395-B Triazolyl aminopyrimidine compounds LILLY CO ELI 2012-06-13 CN disclosed
CN-101679395-A triazolyl aminopyrimidine compounds LILLY CO ELI 2010-03-24 CN disclosed