SCHEMBL27931107

SCHEMBL27931107

CC(CC(C)(C)OC(N)=O)c1ccc(Br)cc1F

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
APLNR P35414 4/20 0.43
AAK1 Q2M2I8 6/20 0.42
DGAT1 O75907 1/20 0.40
ACACB O00763 1/20 0.34
BMP1 P13497 1/20 0.34
FPR2 P25090 2/20 0.33
LMNA P02545 2/20 0.33
NPC1 O15118 1/20 0.33
NFKB1 P19838 1/20 0.33
RAB9A P51151 1/20 0.33
NFKB2 Q00653 1/20 0.33
RELA Q04206 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
ALDH1A1 P00352 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MEN1 O00255 1/20 0.32
MAPT P10636 1/20 0.32
HTT P42858 1/20 0.32
KMT2A Q03164 1/20 0.32
USP30 Q70CQ3 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27931106 1.00 APLNR (0.43) APLNRAAK1DGAT1ACACBBMP1
SCHEMBL27796919 0.82 APLNR (0.37) APLNRAAK1MAPTKMT2A
SCHEMBL28948407 0.79 APLNR (0.46) APLNRAAK1DGAT1ACACBFPR2
SCHEMBL25222547 0.78 ALOX5 (0.43) FPR2LMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL27828808 0.78 ALOX5 (0.43) FPR2LMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL25222546 0.78 ALOX5 (0.43) FPR2LMNASMN1; SMN2ALDH1A1MEN1
SCHEMBL27913119 0.78 APLNR (0.44) APLNRAAK1DGAT1FPR2LMNA
SCHEMBL27498670 0.76 ALDH1A1 (0.37) AAK1ALDH1A1L3MBTL1
SCHEMBL27776366 0.76 HTT (0.40) AAK1NPC1RAB9AALDH1A1MEN1
SCHEMBL27698022 0.76 DGAT1 (0.44) AAK1DGAT1BMP1FPR2MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249727-B Biaryl amide derivatives 霍夫曼-拉罗奇有限公司 2016-08-10 CN disclosed
CN-103249727-A New biaryl amide derivatives HOFFMANN LA ROCHE 2013-08-14 CN disclosed