SCHEMBL27782003

SCHEMBL27782003

N#CC(Br)c1ccccc1F

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TRPA1 O75762 1/20 0.50
IDO1 P14902 2/20 0.36
TDO2 P48775 2/20 0.36
CES2 O00748 1/20 0.36
CES1 P23141 1/20 0.36
ALDH1A1 P00352 4/20 0.35
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
GAA P10253 2/20 0.35
GFER P55789 1/20 0.35
TDP1 Q9NUW8 1/20 0.35
CCR1 P32246 1/20 0.33
MAPT P10636 2/20 0.33
CYP2C9 P11712 2/20 0.33
CYP3A4 P08684 2/20 0.33
NPSR1 Q6W5P4 1/20 0.32
EEF2K O00418 1/20 0.32
CNR2 P34972 2/20 0.32
TSHR P16473 1/20 0.31
ACHE P22303 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28207137 0.78 CES2 (0.40) TRPA1IDO1TDO2CES2CES1
SCHEMBL4910575 0.76 IDO1 (0.37) TRPA1IDO1TDO2CES2CES1
SCHEMBL30145600 0.74 IDO1 (0.40) TRPA1IDO1TDO2CES2CES1
SCHEMBL1023334 0.74 IDO1 (0.40) TRPA1IDO1TDO2CES2CES1
SCHEMBL7868609 0.74 IDO1 (0.40) TRPA1IDO1TDO2CES2CES1
SCHEMBL1628591 0.74 TRPA1 (0.50) TRPA1IDO1TDO2ALDH1A1TDP1
SCHEMBL3495437 0.74 TSHR (0.50) IDO1TDO2CES2CES1ALDH1A1
SCHEMBL1125095 0.74 TRPA1 (0.50) TRPA1ALDH1A1GAACCR1CYP2C9
SCHEMBL9501889 0.74 TRPA1 (0.50) TRPA1ALDH1A1MEN1KMT2AGAA
SCHEMBL2339911 0.74 ALDH1A1 (0.38) IDO1TDO2CES2CES1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-107522634-A Biaryl ureas carboxylic acid derivates or its salt and its production and use 复旦大学 2017-12-29 CN disclosed
CN-102030761-B Prasugrel midbody and preparation method thereof ZHEJIANG PULUO JIAYUAN PHARMACEUTICAL CO LTD 2012-10-10 CN disclosed
CN-102030761-A Prasugrel midbody and preparation method thereof ZHEJIANG PULUO JIAYUAN PHARMACEUTICAL CO LTD 2011-04-27 CN disclosed
CN-101735241-A Prasugrel intermediate and preparation method thereof ZHEJIANG APELOA HOME PHARMACEU 2010-06-16 CN disclosed