Hydralazine

Hydralazine

SCHEMBL2779460

CC(C)=O.NNc1nncc2ccccc12

nearest known ligand 0.81

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 6/20 0.81
RAB9A P51151 5/20 0.81
ALDH1A1 P00352 4/20 0.81
LMNA P02545 3/20 0.81
KDM4E B2RXH2 2/20 0.81
TP53 P04637 2/20 0.81
CYP3A4 P08684 2/20 0.81
GOT1 P17174 2/20 0.81
SMN1; SMN2 Q16637 2/20 0.81
CYP1A2 P05177 2/20 0.81
CYP2D6 P10635 2/20 0.81
MPO P05164 2/20 0.81
MAOA P21397 2/20 0.81
PTGS1 P23219 2/20 0.81
PKM P14618 1/20 0.81
THPO P40225 1/20 0.81
AOX1 Q06278 1/20 0.81
ACOX1 Q15067 1/20 0.81
TDP1 Q9NUW8 3/20 0.78
MAPT P10636 3/20 0.78

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydralazine SCHEMBL2779489 0.92 NPC1 (0.73) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL15140051 0.91 NPC1 (0.71) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL2783124 0.91 NPC1 (0.71) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL3995896 0.90 ALDH1A1 (1.00) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL7810 0.90 ALDH1A1 (1.00) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL2780318 0.88 ALDH1A1 (0.89) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL27864907 0.88 GOT1 (1.00) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL1173534 0.88 GOT1 (1.00) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL36271 0.88 GOT1 (1.00) NPC1RAB9AALDH1A1LMNAKDM4E
Hydralazine SCHEMBL5671747 0.88 NPC1 (0.76) NPC1RAB9AALDH1A1LMNAKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 12 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20130197038-A1 Compositions And Methods For Neovascularization MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2013-08-01 US claimed
US-9446031-B2 Compositions and methods for neovascularization NATIONAL UNIVERSITY OF SINGAPORE (SG) 2016-09-20 US disclosed
US-20130197038-A1 Compositions And Methods For Neovascularization MASSACHUSETTS INSTITUTE OF TECHNOLOGY (US) 2013-08-01 US disclosed
US-7728133-B2 Stable pharmaceutical compositions B&G PARTNERS LLC 2010-06-01 US disclosed
EP-1480649-A4 STABLE PHARMACEUTICAL COMPOSITIONS BARBEAU DONALD L (US) 2006-04-26 EP disclosed
US-20050130975-A1 Stable pharmaceutical compositions B&G PARTNERS LLC 2005-06-16 US disclosed
EP-1480649-A2 STABLE PHARMACEUTICAL COMPOSITIONS Barbeau, Donald L. (US) 2004-12-01 EP disclosed
US-6825196-B2 SUCH AS 1-HYDRAZINOPHTHALAZINE; METAL-FREE BARBEAU PHARMA, INC. 2004-11-30 US disclosed
US-6821974-B2 VASODILATION; HYPOTENSIVE AGENTS; CARDIOVASCULAR DISORDERS BARBEAU PHARMA, INC 2004-11-23 US disclosed
US-20030212272-A1 Stable pharmaceutical compositions B&G PARTNERS LLC 2003-11-13 US disclosed
US-20030199512-A1 Stable pharmaceutical compositions BARBEAU PHARMA INC. 2003-10-23 US disclosed
WO-2003075928-A2 STABLE PHARMACEUTICAL COMPOSITIONS BARBEAU DONALD L (US) 2003-09-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20050130975-A1 Stable pharmaceutical compositions CYP3A7, NR1H2, CYP2B6 NPC1 386/4885RAB9A 1607/4885ALDH1A1 1633/4885
US-20030199512-A1 Stable pharmaceutical compositions H4C1; H4C2; H4C3; H4C4; H4C5; H4C6; H4C8; H4C9; H4C11; H4C12; H4C13; H4C14; H4C15; H4C16, HBZ, HRH1 NPC1 583/4885RAB9A 1189/4885ALDH1A1 446/4885
US-20030212272-A1 Stable pharmaceutical compositions CYP3A7, ARL1, ATXN2L NPC1 441/4885RAB9A 540/4885ALDH1A1 1387/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.