SCHEMBL27811315

SCHEMBL27811315

CNc1cccc(N(C)C(=O)OC(C)(C)C)c1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BRD4 O60885 2/20 0.49
PAX8 Q06710 1/20 0.41
KAT8 Q9H7Z6 1/20 0.38
CREBBP Q92793 1/20 0.38
MEN1 O00255 5/20 0.38
KMT2A Q03164 5/20 0.38
RAB9A P51151 2/20 0.38
NPSR1 Q6W5P4 1/20 0.38
ALDH1A1 P00352 3/20 0.37
MAPK1 P28482 2/20 0.37
HTT P42858 1/20 0.37
BCHE P06276 1/20 0.36
ACHE P22303 1/20 0.36
USP30 Q70CQ3 1/20 0.35
MAPT P10636 2/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
USP2 O75604 1/20 0.35
LMNA P02545 1/20 0.35
GAA P10253 1/20 0.35
ALOX15 P16050 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL18513515 0.86 MEN1 (0.49) BRD4MEN1KMT2ARAB9AALDH1A1
SCHEMBL2450799 0.82 L3MBTL1 (0.52) BRD4RAB9ANPSR1MAPTSMN1; SMN2
SCHEMBL8749479 0.81 PAX8 (0.47) BRD4PAX8KAT8CREBBPMEN1
SCHEMBL10210873 0.80 BRD4 (0.52) BRD4PAX8MAPK1MAPTSMN1; SMN2
SCHEMBL30504285 0.80 BRD4 (0.62) BRD4PAX8KAT8CREBBPMEN1
SCHEMBL3910121 0.79 BRD4 (0.51) BRD4PAX8KAT8CREBBPMEN1
SCHEMBL14065550 0.79 BRD4 (0.51) BRD4PAX8KAT8CREBBPMEN1
SCHEMBL67115 0.79 BRD4 (0.51) BRD4PAX8CREBBPMEN1KMT2A
SCHEMBL30013638 0.79 BRD4 (0.51) BRD4PAX8CREBBPMEN1KMT2A
SCHEMBL30455057 0.79 HTR3E (0.51) BRD4PAX8KMT2ANPSR1ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102740847-A Heteroaryl compounds and uses thereof AVILA THERAPEUTICS INC 2012-10-17 CN disclosed
CN-102083800-A Heteroaryl compounds and uses thereof AVILA THERAPEUTICS AND USES TH 2011-06-01 CN disclosed