SCHEMBL27823919

SCHEMBL27823919

COc1c(Br)cccc1C(C)C(=O)C(C)c1cccc(Br)c1OC

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2C9 P11712 2/20 0.38
CYP2C19 P33261 2/20 0.38
MEN1 O00255 2/20 0.37
KMT2A Q03164 2/20 0.37
HTT P42858 2/20 0.36
TSHR P16473 1/20 0.36
APOBEC3A P31941 1/20 0.36
APOBEC3G Q9HC16 1/20 0.36
LPAR1 Q92633 2/20 0.35
CYP1A2 P05177 1/20 0.35
CYP3A4 P08684 1/20 0.35
TUBB4A P04350 2/20 0.35
TUBB P07437 2/20 0.35
TUBA3C P0DPH7 2/20 0.35
TUBA1B P68363 2/20 0.35
TUBA4A P68366 2/20 0.35
TUBB4B P68371 2/20 0.35
TUBB3 Q13509 2/20 0.35
TUBB2A Q13885 2/20 0.35
TUBB8 Q3ZCM7 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2899680 0.88 PTGS2 (0.46) CYP2C9CYP2C19MEN1KMT2ATSHR
SCHEMBL32681778 0.80 KMT2A (0.36) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL3065896 0.80 KMT2A (0.36) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL29731059 0.80 KMT2A (0.36) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL1680252 0.80 KMT2A (0.36) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL618635 0.80 GABRA1 (0.41) CYP2C9CYP2C19MEN1KMT2ATSHR
SCHEMBL23526320 0.78 HTT (0.46) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL28880510 0.78 HTT (0.39) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL30014041 0.78 HTT (0.46) CYP2C9CYP2C19MEN1KMT2AHTT
SCHEMBL23526323 0.78 HTT (0.46) CYP2C9CYP2C19MEN1KMT2AHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-101981034-B Triazolopyridazines as PAR1 inhibitors, their preparation and their use for producing medicaments SANOFI AVENTIS 2013-08-14 CN disclosed
CN-101981034-A Triazolopyridazines as PAR1 inhibitors, their preparation and their use as medicaments SANOFI AVENTIS 2011-02-23 CN disclosed