SCHEMBL27877036

SCHEMBL27877036

Cc1cccc(C(=O)Nc2nnc(S)s2)c1

nearest known ligand 0.62

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.62
KMT2A Q03164 7/20 0.61
MAPT P10636 7/20 0.61
MEN1 O00255 6/20 0.61
NPC1 O15118 2/20 0.57
RAB9A P51151 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
SCD O00767 1/20 0.57
KDM4E B2RXH2 1/20 0.57
ALDH1A1 P00352 1/20 0.56
GAA P10253 1/20 0.56
ALOX15 P16050 1/20 0.56
TSHR P16473 1/20 0.56
THRB P10828 1/20 0.56
G6PD P11413 1/20 0.55
TP53 P04637 2/20 0.54
KCNK3 O14649 1/20 0.54
KCNH2 Q12809 1/20 0.54
KCNK9 Q9NPC2 1/20 0.54
RXFP1 Q9HBX9 2/20 0.54

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8556554 0.86 KMT2A (0.75) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL27877118 0.85 SMN1; SMN2 (0.51) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL2664519 0.82 SMN1; SMN2 (0.67) KMT2AMAPTMEN1NPC1RAB9A
SCHEMBL8556694 0.81 KMT2A (0.69) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL18762149 0.79 KMT2A (0.73) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL27860322 0.78 TP53 (0.55) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL8554413 0.78 LMNA (0.65) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL17318577 0.76 KDM4E (0.73) KMT2AMAPTMEN1NPC1RAB9A
SCHEMBL8554147 0.76 LMNA (0.65) LMNAKMT2AMAPTMEN1NPC1
SCHEMBL8559786 0.76 RAB9A (0.74) LMNAKMT2AMAPTMEN1NPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102532126-B 2-substituted-4-chloro-5-[5-subtsituted amino-2-(1,3,4-thiadiazole)-sulfydryl]-3(2H)- pyridazinone derivatives, and preparation method and application thereof UNIV GUIZHOU 2014-06-18 CN disclosed
CN-102532126-A 2-substituted-4-chloro-5-[5-subtsituted amino-2-(1,3,4-thiadiazole)-sulfydryl]-3(2H)- pyridazinone derivatives, and preparation method and application thereof UNIV GUIZHOU 2012-07-04 CN disclosed