SCHEMBL8554147

SCHEMBL8554147

Cc1cccc(C(=O)Nc2nncs2)c1

nearest known ligand 0.65

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
LMNA P02545 1/20 0.65
AQP4 P55087 1/20 0.60
KMT2A Q03164 4/20 0.57
MEN1 O00255 3/20 0.57
KDM4E B2RXH2 1/20 0.56
RAB9A P51151 2/20 0.55
SCD O00767 1/20 0.55
NPC1 O15118 1/20 0.55
SMN1; SMN2 Q16637 1/20 0.55
KCNK3 O14649 1/20 0.55
KCNH2 Q12809 1/20 0.55
KCNK9 Q9NPC2 1/20 0.55
NT5E P21589 1/20 0.54
MAPT P10636 2/20 0.53
ALDH1A1 P00352 1/20 0.52
HPGD P15428 1/20 0.52
HSD17B10 Q99714 1/20 0.52
GRM5 P41594 1/20 0.52
TP53 P04637 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7348856 0.83 LMNA (0.62) LMNAAQP4KMT2AMEN1KDM4E
SCHEMBL3379803 0.82 AQP4 (0.70) LMNAAQP4KMT2AMEN1KDM4E
SCHEMBL9963857 0.79 KDM4E (0.61) LMNAAQP4KMT2AMEN1KDM4E
SCHEMBL8556554 0.78 KMT2A (0.75) LMNAKMT2AMEN1KDM4ERAB9A
SCHEMBL8555330 0.77 TP53 (0.70) LMNAKMT2AMEN1KDM4ERAB9A
SCHEMBL8560618 0.77 GCK (0.79) LMNARAB9ANPC1SMN1; SMN2MAPT
SCHEMBL8157997 0.77 RAB9A (0.63) LMNAAQP4KMT2AMEN1KDM4E
SCHEMBL3893137 0.77 RAB9A (0.60) LMNAAQP4KMT2AMEN1KDM4E
SCHEMBL27877036 0.76 LMNA (0.62) LMNAKMT2AMEN1KDM4ERAB9A
SCHEMBL8554959 0.74 RAB9A (0.70) LMNAKMT2AMEN1KDM4ERAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP claimed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US claimed
EP-0815108-A1 CYCLIC UREA HIV PROTEASE INHIBITORS THE DU PONT MERCK PHARMACEUTICAL COMPANY (US) 1998-01-07 EP disclosed
US-5683999-A Cyclic urea HIV protease inhibitors THE DUPONT MERCK PHARMACEUTICAL COMPANY (US) 1997-11-04 US disclosed