SCHEMBL2788286

SCHEMBL2788286

CC(=O)c1ccc(NC(=O)NSc2noc3ccccc23)cc1

nearest known ligand 0.61

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HIF1A Q16665 6/20 0.61
RAB9A P51151 7/20 0.49
NPC1 O15118 6/20 0.49
MAPT P10636 5/20 0.49
SMN1; SMN2 Q16637 4/20 0.49
TAAR1 Q96RJ0 1/20 0.49
KMT2A Q03164 4/20 0.46
KDM4E B2RXH2 2/20 0.43
MEN1 O00255 2/20 0.42
PIK3R1 P27986 1/20 0.42
PIK3CA P42336 1/20 0.42
MTOR P42345 1/20 0.42
HTT P42858 1/20 0.42
NLRP1 Q9C000 1/20 0.42
ALDH1A1 P00352 1/20 0.41
TP53 P04637 1/20 0.41
CA12 O43570 1/20 0.41
CA1 P00915 1/20 0.41
CA2 P00918 1/20 0.41
CA9 Q16790 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2785339 0.81 HIF1A (0.45) HIF1ARAB9ANPC1MAPTSMN1; SMN2
SCHEMBL2768846 0.73 HIF1A (0.64) HIF1ARAB9ANPC1MAPTSMN1; SMN2
SCHEMBL2786818 0.73 RAB9A (0.41) HIF1ARAB9ANPC1MAPTSMN1; SMN2
SCHEMBL1719786 0.68 RAB9A (1.00) RAB9ANPC1MAPTSMN1; SMN2TAAR1
SCHEMBL3633396 0.67 NPC1 (0.84) RAB9ANPC1MAPTSMN1; SMN2TAAR1
SCHEMBL2785931 0.67 GHSR (0.47) RAB9ANPC1MAPTKMT2AMEN1
SCHEMBL2785316 0.67 TP53 (0.52) HIF1AMAPTSMN1; SMN2TP53
SCHEMBL2788190 0.66 SMN1; SMN2 (0.55) HIF1ARAB9ANPC1MAPTSMN1; SMN2
SCHEMBL2785576 0.66 SMN1; SMN2 (0.48) HIF1ARAB9ANPC1MAPTSMN1; SMN2
SCHEMBL23069083 0.65 RAB9A (0.86) RAB9ANPC1MAPTSMN1; SMN2TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1881967-B1 SUBSTITUTED BENZO(D)ISOXAZOL-3-YL AMINE COMPOUNDS AS ANALGESICS GRUENENTHAL GMBH (DE) 2010-04-28 EP claimed