SCHEMBL27895604

SCHEMBL27895604

CC(=O)Oc1nc(N)ccc1C

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS3 P29474 1/20 0.45
NOS1 P29475 1/20 0.45
NOS2 P35228 1/20 0.45
GABRP O00591 4/20 0.42
GABRD O14764 4/20 0.42
GABRA1 P14867 4/20 0.42
GABRB1 P18505 4/20 0.42
GABRG2 P18507 4/20 0.42
GABRB3 P28472 4/20 0.42
GABRA5 P31644 4/20 0.42
GABRA3 P34903 4/20 0.42
GABRA2 P47869 4/20 0.42
GABRB2 P47870 4/20 0.42
GABRA4 P48169 4/20 0.42
GABRE P78334 4/20 0.42
GABRA6 Q16445 4/20 0.42
GABRG1 Q8N1C3 4/20 0.42
GABRG3 Q99928 4/20 0.42
GABRQ Q9UN88 4/20 0.42
LMNA P02545 3/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27703245 0.81 LMNA (0.38) LMNAACHEALOX5KDM4EHTT
SCHEMBL27570781 0.81 LMNA (0.41) LMNAACHEALOX5KDM4EHTT
SCHEMBL27789443 0.80 GABRP (0.37) NOS3NOS1NOS2GABRPGABRD
SCHEMBL2829068 0.74 GABRP (0.50) NOS3NOS1NOS2GABRPGABRD
SCHEMBL15544743 0.74 NOS2 (0.54) NOS3NOS1NOS2GABRPGABRD
SCHEMBL16834762 0.74 LMNA (0.39) LMNAACHEALOX5KDM4ETP53
SCHEMBL15544912 0.74 KDM4E (0.42) LMNAKDM4ETSHRALDH1A1HPGD
SCHEMBL27850349 0.70 GRM5 (0.40) NOS3NOS2LMNAALOX5KDM4E
SCHEMBL27878809 0.70 ALOX5 (0.35) GABRPGABRDGABRA1GABRB1GABRG2
SCHEMBL28783444 0.69 ALOX5 (0.36) LMNAALOX5KDM4EGAAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102762561-A Gamma secretase modulaters HOFFMANN LA ROCHE 2012-10-31 CN disclosed