SCHEMBL2790403

SCHEMBL2790403

COCCCn1c(C2CCCN(C(=O)CC(Cc3ccc(NC(=O)c4cc(C)nn4C)cc3)NC(=O)OC(C)(C)C)C2)c(C)c2cccc(F)c21

nearest known ligand 0.32

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
PABPC1 P11940 1/20 0.32
CYP2D6 P10635 2/20 0.31
ALDH1A1 P00352 1/20 0.31
LMNA P02545 1/20 0.31
CYP3A4 P08684 1/20 0.31
CYP2C9 P11712 1/20 0.31
CYP2C19 P33261 1/20 0.31
EEF2K O00418 1/20 0.31
CCR3 P51677 1/20 0.31
STING1 Q86WV6 2/20 0.31
KLK5 Q9Y337 1/20 0.31
PIN1 Q13526 1/20 0.31
ATM Q13315 1/20 0.31
USP1 O94782 1/20 0.30
GFER P55789 1/20 0.30
MAPK1 P28482 1/20 0.30
PADI4 Q9UM07 1/20 0.30
BACE1 P56817 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2790406 1.00 PABPC1 (0.32) PABPC1CYP2D6ALDH1A1LMNACYP3A4
SCHEMBL2880505 0.95 STING1 (0.36) CYP2D6ALDH1A1LMNACYP3A4CYP2C9
SCHEMBL2880502 0.95 STING1 (0.36) CYP2D6ALDH1A1LMNACYP3A4CYP2C9
SCHEMBL2791715 0.94 ALDH1A1 (0.33) PABPC1CYP2D6ALDH1A1LMNACYP3A4
SCHEMBL2791712 0.94 ALDH1A1 (0.33) PABPC1CYP2D6ALDH1A1LMNACYP3A4
SCHEMBL7900833 0.92 PABPC1 (0.34) PABPC1CYP2D6ALDH1A1CCR3KLK5
SCHEMBL2791534 0.89 MMP13 (0.34) PABPC1CYP2D6ALDH1A1LMNACYP3A4
SCHEMBL7899253 0.89 PABPC1 (0.32) PABPC1CYP2D6ALDH1A1LMNACYP3A4
SCHEMBL2788011 0.89 DPP4 (0.33) CYP2D6CCR3PIN1ATMUSP1
SCHEMBL2788008 0.89 DPP4 (0.33) CYP2D6CCR3PIN1ATMUSP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed