SCHEMBL7900833

SCHEMBL7900833

COCCCn1c(C2CCCN(C(=O)C[C@@H](Cc3ccc(NC(=O)c4ccnn4C)cc3)NC(=O)OC(C)(C)C)C2)c(C)c2cccc(F)c21

nearest known ligand 0.34

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
PABPC1 P11940 1/20 0.34
CMA1 P23946 2/20 0.31
KLK5 Q9Y337 1/20 0.31
PTPN1 P18031 2/20 0.30
ALDH1A1 P00352 1/20 0.30
TSHR P16473 1/20 0.30
KMT2A Q03164 1/20 0.30
CYP2D6 P10635 1/20 0.30
CCR3 P51677 1/20 0.30
ACE P12821 1/20 0.30
CCKAR P32238 2/20 0.30
CCKBR P32239 2/20 0.30
HRH2 P25021 1/20 0.30
HRH1 P35367 1/20 0.30
IL17A Q16552 1/20 0.30
ATM Q13315 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2790406 0.92 PABPC1 (0.32) PABPC1KLK5ALDH1A1CYP2D6CCR3
SCHEMBL2790403 0.92 PABPC1 (0.32) PABPC1KLK5ALDH1A1CYP2D6CCR3
SCHEMBL2791715 0.90 ALDH1A1 (0.33) PABPC1ALDH1A1CYP2D6CCR3
SCHEMBL2791712 0.90 ALDH1A1 (0.33) PABPC1ALDH1A1CYP2D6CCR3
SCHEMBL2880502 0.90 STING1 (0.36) ALDH1A1CYP2D6
SCHEMBL2880505 0.90 STING1 (0.36) ALDH1A1CYP2D6
SCHEMBL7898847 0.90 MMP13 (0.35) PABPC1KLK5ALDH1A1KMT2ACYP2D6
SCHEMBL2791534 0.89 MMP13 (0.34) PABPC1KLK5ALDH1A1CYP2D6
SCHEMBL7897783 0.89 PABPC1 (0.33) PABPC1KLK5PTPN1
SCHEMBL7901258 0.89 PABPC1 (0.33) PABPC1KLK5HRH2HRH1ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed