SCHEMBL2880505

SCHEMBL2880505

CCn1nc(C)cc1C(=O)Nc1ccc(C[C@H](CC(=O)N2CCCC(c3c(C)c4cccc(F)c4n3CCCOC)C2)NC(=O)OC(C)(C)C)cc1

nearest known ligand 0.36

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
STING1 Q86WV6 16/20 0.36
CYP3A4 P08684 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GFER P55789 1/20 0.32
ALDH1A1 P00352 1/20 0.32
LMNA P02545 1/20 0.32
CYP2D6 P10635 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2880502 1.00 STING1 (0.36) STING1CYP3A4KDM4EGFERALDH1A1
SCHEMBL2790406 0.95 PABPC1 (0.32) STING1CYP3A4GFERALDH1A1LMNA
SCHEMBL2790403 0.95 PABPC1 (0.32) STING1CYP3A4GFERALDH1A1LMNA
SCHEMBL2791715 0.91 ALDH1A1 (0.33) CYP3A4GFERALDH1A1LMNACYP2D6
SCHEMBL2791712 0.91 ALDH1A1 (0.33) CYP3A4GFERALDH1A1LMNACYP2D6
SCHEMBL7900833 0.90 PABPC1 (0.34) ALDH1A1CYP2D6
SCHEMBL2788172 0.89 STING1 (0.36) STING1KDM4EGFER
SCHEMBL2788169 0.89 STING1 (0.36) STING1KDM4EGFER
SCHEMBL2791534 0.89 MMP13 (0.34) CYP3A4ALDH1A1LMNACYP2D6CYP2C9
SCHEMBL7898847 0.88 MMP13 (0.35) CYP3A4ALDH1A1LMNACYP2D6CYP2C9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed
WO-2010111634-A2 RENIN INHIBITORS TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-09-30 WO disclosed