SCHEMBL27913626

SCHEMBL27913626

Cc1cc(C(=O)NCc2cc(F)cc(C(F)(F)F)c2)ccn1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NAMPT P43490 1/20 0.52
MLYCD O95822 1/20 0.51
TACR1 P25103 3/20 0.51
KDM1A O60341 1/20 0.49
HDAC1 Q13547 1/20 0.49
EGLN1 Q9GZT9 1/20 0.48
WDR5 P61964 2/20 0.48
ALDH1A1 P00352 5/20 0.48
KDM4E B2RXH2 4/20 0.48
HPGD P15428 4/20 0.48
CYP3A4 P08684 3/20 0.48
CYP2D6 P10635 2/20 0.48
CYP1A2 P05177 1/20 0.48
CYP2C9 P11712 1/20 0.48
CYP2C19 P33261 1/20 0.48
AURKA O14965 1/20 0.46
HTT P42858 2/20 0.46
LMNA P02545 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
PSEN1 P49768 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27931807 0.85 MLYCD (0.62) MLYCDHDAC1HPGDCYP3A4CYP2D6
SCHEMBL2718344 0.84 NAMPT (0.51) NAMPTMLYCDTACR1KDM1AHDAC1
SCHEMBL27931803 0.84 L3MBTL1 (0.62) NAMPTMLYCDKDM1AHDAC1EGLN1
SCHEMBL2715156 0.83 NAMPT (0.49) NAMPTMLYCDTACR1KDM1AHDAC1
SCHEMBL28094014 0.82 VNN1 (0.45) TACR1WDR5ALDH1A1CYP3A4CYP2D6
SCHEMBL2715620 0.82 SCN9A (0.56) NAMPTMLYCDTACR1KDM1AHDAC1
SCHEMBL27913768 0.80 MMP13 (0.50) NAMPTMLYCDTACR1ALDH1A1CYP3A4
SCHEMBL2717667 0.80 GSK3B (0.53) NAMPT
SCHEMBL6253464 0.79 MLYCD (0.60) MLYCDTACR1KDM1AHDAC1ALDH1A1
SCHEMBL27913563 0.79 DDR1 (0.47) KDM1AHDAC1WDR5LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN claimed
CN-103249721-A Arylamine Derivatives as TTX-S Blockers RAQUALIA PHARMA INC 2013-08-14 CN disclosed