SCHEMBL279238

SCHEMBL279238

COCc1nccc(Oc2ccc3c(C(=O)Nc4ccccc4)cccc3c2)n1

nearest known ligand 0.70

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
KDR P35968 20/20 0.70
RET P07949 2/20 0.63
FLT1 P17948 2/20 0.63
PDGFRB P09619 1/20 0.56
KIT P10721 1/20 0.56
FLT4 P35916 1/20 0.56

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2470527 0.95 KDR (0.66) KDRRETFLT1PDGFRBKIT
SCHEMBL2468881 0.91 KDR (0.68) KDRRETFLT1PDGFRBKIT
SCHEMBL2469884 0.89 KDR (0.63) KDRRETFLT1PDGFRBKIT
SCHEMBL2467345 0.89 KDR (0.56) KDRRETFLT1PDGFRBKIT
SCHEMBL278839 0.89 KDR (0.74) KDRRETFLT1PDGFRBKIT
SCHEMBL2473044 0.89 KDR (0.57) KDRRETFLT1PDGFRBKIT
SCHEMBL2467550 0.89 KDR (0.74) KDRRETFLT1PDGFRBKIT
SCHEMBL2469406 0.88 KDR (0.59) KDRRETFLT1PDGFRBKIT
SCHEMBL273334 0.88 KDR (0.55) KDRRETFLT1PDGFRBKIT
SCHEMBL3595046 0.87 KDR (0.51) KDRRETFLT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20120122857-A1 HETEROBICYCLIC CARBOXAMIDES AS INHIBITORS FOR KINASES NOVARTIS AG (CH) 2012-05-17 US disclosed
US-8133886-B2 Heterobicyclic carboxamides as inhibitors for kinases NOVARTIS AG (CH) 2012-03-13 US disclosed
US-20100029626-A1 Cyclic sulfones useful as mitochondrial sodium-calcium exchangers NOVARTIS AG (CH) 2010-02-04 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20100029626-A1 Cyclic sulfones useful as mitochondrial sodium-calcium exchangers SLC8B1, MCU, GLS KDR 3083/4885RET 2287/4885FLT1 2466/4885
US-20120122857-A1 HETEROBICYCLIC CARBOXAMIDES AS INHIBITORS FOR KINASES MAP3K20, PHKG1, PHKG2 KDR 1319/4885RET 322/4885FLT1 1353/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.