SCHEMBL27972717

SCHEMBL27972717

O=C1CC(c2ccccc2)C(Cc2ccccc2Cl)N1

nearest known ligand 0.43

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
CES2 O00748 2/20 0.39
NR3C1 P04150 3/20 0.38
LMNA P02545 3/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
CMA1 P23946 1/20 0.37
P2RX7 Q99572 1/20 0.37
ALDH1A1 P00352 3/20 0.37
SLC6A3 Q01959 1/20 0.37
NR3C2 P08235 1/20 0.36
DAO P14920 1/20 0.35
KDM4E B2RXH2 1/20 0.35
MAPT P10636 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17184797 0.74 KDM1A (0.39) KDM1ANPSR1LMNAMEN1KMT2A
SCHEMBL6985693 0.73 ITGB1 (0.49) KDM1ANPSR1LMNAALDH1A1
SCHEMBL6990768 0.73 NPSR1 (0.44) NPSR1LMNAALDH1A1KDM4EMAPT
SCHEMBL5481415 0.71 NPSR1 (0.45) KDM1ANPSR1LMNAALDH1A1KDM4E
SCHEMBL7117751 0.67 DRD2 (0.42) LMNAALDH1A1SLC6A3KDM4E
SCHEMBL7117749 0.67 DRD2 (0.42) LMNAALDH1A1SLC6A3KDM4E
SCHEMBL11355593 0.67 CMA1 (0.45) CES2MEN1KMT2ACMA1ALDH1A1
SCHEMBL29049348 0.67 FFAR1 (0.46) NPSR1LMNACMA1ALDH1A1MAPT
SCHEMBL17523286 0.67 SLC6A3 (0.41) NPSR1MEN1KMT2AALDH1A1SLC6A3
SCHEMBL1901694 0.66 ALDH1A1 (0.48) NPSR1LMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103877080-B 4,5-bis-replaces-medicinal usage of 2-Pyrrolidone compound Key Laboratory of natural product chemistry, Chinese Academy of Sciences, Guizhou Province (CN) 2016-01-27 CN claimed
CN-103877080-A New use of 4, 5-disubstituted-2-pyrrolidone compound KEY LAB OF CHEMISTRY NATURAL PRODUCTS OF GUIZHOU PROVINCE AND CHINESE ACADEMY 2014-06-25 CN claimed
CN-103877080-B 4,5-bis-replaces-medicinal usage of 2-Pyrrolidone compound Key Laboratory of natural product chemistry, Chinese Academy of Sciences, Guizhou Province (CN) 2016-01-27 CN disclosed
CN-103877080-A New use of 4, 5-disubstituted-2-pyrrolidone compound KEY LAB OF CHEMISTRY NATURAL PRODUCTS OF GUIZHOU PROVINCE AND CHINESE ACADEMY 2014-06-25 CN disclosed