SCHEMBL27995719

SCHEMBL27995719

CC(Br)c1ccc2[nH]ncc2c1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 5/20 0.55
METAP2 P50579 2/20 0.55
CSNK2A1 P68400 1/20 0.55
ROCK2 O75116 6/20 0.50
ROCK1 Q13464 3/20 0.50
MAPT P10636 2/20 0.50
KDM4E B2RXH2 1/20 0.50
MEN1 O00255 1/20 0.50
ALDH1A1 P00352 1/20 0.50
GAA P10253 1/20 0.50
HPGD P15428 1/20 0.50
RAB9A P51151 1/20 0.50
KMT2A Q03164 1/20 0.50
HIF1A Q16665 1/20 0.50
TDP1 Q9NUW8 1/20 0.50
TRPA1 O75762 6/20 0.48
GSK3B P49841 3/20 0.46
CLK1 P49759 2/20 0.46
DYRK1A Q13627 2/20 0.46
DYRK3 O43781 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL15673661 0.86 NOS1 (0.56) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL6181437 0.86 NOS1 (0.55) NOS1METAP2CSNK2A1MAPTKDM4E
SCHEMBL84462 0.85 TRPA1 (0.54) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL1754871 0.82 ROCK2 (0.55) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL263567 0.82 ROCK2 (0.55) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL20841219 0.82 NOS1 (0.55) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL30074251 0.82 ROCK2 (0.50) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL22079235 0.82 ROCK2 (0.55) NOS1METAP2CSNK2A1ROCK2ROCK1
SCHEMBL29520764 0.81 TRPA1 (0.54) NOS1METAP2CSNK2A1ROCK2ROCK1
Hydrochloric Acid SCHEMBL29915566 0.81 ROCK2 (0.53) NOS1METAP2CSNK2A1ROCK2ROCK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105358559-A Pyrrolopyridine or pyrazolopyridine derivative HOFFMANN LA ROCHE 2016-02-24 CN disclosed
CN-104884451-A Pyridinone and pyridazinone derivatives ABBVIE INC 2015-09-02 CN disclosed
CN-104718201-A Pyridinone and pyridazinone derivatives ABBVIE INC 2015-06-17 CN disclosed
CN-104379573-A Isoindolone derivatives ABBVIE INC 2015-02-25 CN disclosed
CN-104334526-A Isoindolone derivatives ABBVIE INC 2015-02-04 CN disclosed