SCHEMBL28017381

SCHEMBL28017381

CN(C(=O)CNC(=O)OC(C)(C)C)c1cc(-c2ccc(C(F)(F)F)cc2)ncn1

nearest known ligand 0.40

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
AURKB Q96GD4 1/20 0.40
AAK1 Q2M2I8 6/20 0.40
P2RY14 Q15391 4/20 0.39
FAAH O00519 1/20 0.39
ABL1 P00519 2/20 0.39
BCR P11274 2/20 0.39
ADORA3 P0DMS8 1/20 0.36
KCNH2 Q12809 1/20 0.36
TRPV1 Q8NER1 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL16894189 0.83 CACNA1G (0.38) AAK1FAAHKCNH2TRPV1
SCHEMBL28017384 0.82 ALDH1A1 (0.38) AAK1FAAHABL1BCRADORA3
SCHEMBL16894276 0.80 AAK1 (0.36) AAK1FAAHKCNH2TRPV1
SCHEMBL16965653 0.74 KMT2A (0.40) FAAHABL1BCRADORA3KCNH2
SCHEMBL893757 0.72 HDAC1 (0.53) P2RY14TRPV1
SCHEMBL2585523 0.72 TBK1 (0.46)
SCHEMBL18068201 0.71 KDM1A (0.42) AAK1P2RY14ADORA3
SCHEMBL16894191 0.71 TRPA1 (0.47) AAK1TRPV1
SCHEMBL17979180 0.69 HDAC1 (0.43) AAK1P2RY14ADORA3
SCHEMBL4704775 0.68 CYP17A1 (0.43)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104684899-B Substituted sulfonamide compounds 霍夫曼-拉罗奇有限公司 2017-07-04 CN disclosed
CN-104684899-A Substituted sulfonamide compounds HOFFMANN LA ROCHE 2015-06-03 CN disclosed