SCHEMBL28019667

SCHEMBL28019667

O=C(OC1CCCCC1)N1CCC(c2ccc(OCc3ccccc3)cc2OCc2ccccc2)C1

nearest known ligand 0.48

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
GHSR Q92847 1/20 0.48
PDE4B Q07343 2/20 0.47
HRH3 Q9Y5N1 4/20 0.44
CYP2D6 P10635 2/20 0.43
GRIN1 Q05586 2/20 0.43
GRIN2B Q13224 2/20 0.43
F2 P00734 1/20 0.43
PRSS1 P07477 1/20 0.43
SGMS2 Q8NHU3 1/20 0.41
SPHK1 Q9NYA1 1/20 0.41
KDM2B Q8NHM5 1/20 0.41
SPHK2 Q9NRA0 1/20 0.41
OPRD1 P41143 1/20 0.41
OPRK1 P41145 1/20 0.41
TP53 P04637 1/20 0.40
SMN1; SMN2 Q16637 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28019664 0.87 GRIN1 (0.48) HRH3CYP2D6GRIN1GRIN2BSPHK1
SCHEMBL2476770 0.84 YAP1 (0.52) GHSR
SCHEMBL2478075 0.83 SGMS2 (0.50) HRH3SGMS2SMN1; SMN2
SCHEMBL2475047 0.83 PDE4B (0.46) GHSRPDE4BGRIN1GRIN2BKDM2B
SCHEMBL16564510 0.82 HTR1A (0.48) HRH3GRIN1GRIN2BSPHK1SPHK2
SCHEMBL2475650 0.80 ALDH1A1 (0.56) SMN1; SMN2
SCHEMBL3354512 0.79 ALDH1A1 (0.57) SPHK1SPHK2TP53SMN1; SMN2
SCHEMBL3356183 0.77 ALDH1A1 (0.54) SPHK1SPHK2TP53SMN1; SMN2
SCHEMBL2478613 0.76 GHSR (0.49) GHSRKDM2B
SCHEMBL13504469 0.75 GRIN1 (0.43) HRH3CYP2D6GRIN1GRIN2BSPHK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104666299-A 4-(azacycloalkyl)benzene-1,3-diol compounds as tyrosinase inhibitors, process for the preparation thereof and use thereof GALDERMA RES & DEV 2015-06-03 CN disclosed