SCHEMBL4729623

SCHEMBL4729623

CCCc1cncc2ccc(C(=O)NN)nc12

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.44
GAA P10253 2/20 0.43
ALDH1A1 P00352 1/20 0.43
MAPT P10636 1/20 0.43
CCNC P24863 7/20 0.40
CDK8 P49336 7/20 0.40
KDM4E B2RXH2 2/20 0.35
HDAC3 O15379 1/20 0.34
HDAC1 Q13547 1/20 0.34
HDAC2 Q92769 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
MCL1 Q07820 1/20 0.33
L3MBTL1 Q9Y468 1/20 0.33
MPO P05164 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP3A4 P08684 1/20 0.33
ADORA3 P0DMS8 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2A6 P11509 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4728279 0.77 ALDH1A1 (0.47) P2RX7GAAALDH1A1MAPTCCNC
SCHEMBL4729625 0.76 P2RX7 (0.45) P2RX7GAAALDH1A1MAPTCCNC
SCHEMBL4730799 0.76 P2RX7 (0.45) P2RX7GAAALDH1A1MAPTCCNC
SCHEMBL28024769 0.74 CCNC (0.44) ALDH1A1CCNCCDK8
SCHEMBL9000752 0.73 MAPT (0.61) P2RX7GAAALDH1A1MAPTKDM4E
SCHEMBL28024317 0.72 CCNC (0.48) CCNCCDK8KMT2AADORA3
SCHEMBL28821388 0.70 CCNC (0.44) CCNCCDK8
SCHEMBL15741758 0.68 CCNC (0.46) CCNCCDK8L3MBTL1
SCHEMBL14287007 0.68 SMYD3 (0.40) CCNCCDK8
SCHEMBL4729283 0.67 ALDH1A1 (0.63) P2RX7GAAALDH1A1MAPTKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith D SIDOCKY NEIL R 2008-10-02 US disclosed
WO-2008036308-A2 AMINO-SUBSTITUTED HETEROCYCLES, COMPOSITIONS THEREOF, AND METHODS OF TREATMENT THEREWITH SIGNAL PHARMACEUTICALS, LLC (US) 2008-03-27 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20080242694-A1 Amino-substituted heterocycles, compositions thereof, and methods of treatment therewith JAK2, CHEK2, MTOR P2RX7 1319/4885GAA 2251/4885ALDH1A1 1752/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.