SCHEMBL28025183

SCHEMBL28025183

N#Cc1ncccc1N1CCOCC1Br

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNMA1 Q12791 1/20 0.36
GRM1 Q13255 2/20 0.35
CYP3A4 P08684 1/20 0.35
CYP2D6 P10635 1/20 0.35
PDE4D Q08499 2/20 0.33
USP30 Q70CQ3 1/20 0.33
NPC1 O15118 1/20 0.33
KDM4E B2RXH2 4/20 0.33
MTOR P42345 4/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
HSD17B10 Q99714 3/20 0.33
PIK3C3 Q8NEB9 1/20 0.33
NUDT1 P36639 1/20 0.32
MAPK1 P28482 1/20 0.32
LRRK2 Q5S007 1/20 0.32
LMNA P02545 1/20 0.32
CYP11B1 P15538 1/20 0.32
ATR Q13535 2/20 0.31
ATRIP Q8WXE1 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28024746 0.80 PIK3CD (0.36) PDE4DNPC1KDM4EMTORALDH1A1
SCHEMBL2084217 0.76 ALDH1A1 (0.51) KCNMA1GRM1CYP3A4CYP2D6PDE4D
SCHEMBL27866878 0.71 GRIN2D (0.40) KDM4EMTORPIK3C3ATRATRIP
SCHEMBL28025174 0.68 CHRNB2 (0.41) MTORPIK3C3MAPK1ATRATRIP
SCHEMBL30307674 0.67 KDM4E (0.47) KCNMA1GRM1CYP3A4CYP2D6KDM4E
SCHEMBL21722473 0.67 KDM4E (0.47) KCNMA1GRM1CYP3A4CYP2D6KDM4E
SCHEMBL21722525 0.67 GRM1 (0.45) KCNMA1GRM1CYP3A4CYP2D6KDM4E
SCHEMBL30206003 0.67 AKR1C3 (0.46) KDM4EALDH1A1HPGDHSD17B10MAPK1
SCHEMBL2084707 0.66 KCNMA1 (0.48) KCNMA1GRM1CYP3A4CYP2D6NPC1
SCHEMBL28025203 0.66 ATR (0.35) KDM4EALDH1A1PIK3C3ATRATRIP

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143209-A Biaryl amide compounds as kinase inhibitors NOVARTIS AG 2015-12-09 CN disclosed