SCHEMBL28024746

SCHEMBL28024746

Oc1ncccc1N1CCOCC1Br

nearest known ligand 0.36

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
PIK3CD O00329 1/20 0.36
PIK3CA P42336 1/20 0.36
NUDT1 P36639 1/20 0.34
NPC1 O15118 2/20 0.33
RAB9A P51151 2/20 0.33
L3MBTL1 Q9Y468 2/20 0.33
METAP2 P50579 1/20 0.33
PAX8 Q06710 1/20 0.33
PDE4D Q08499 1/20 0.33
ATR Q13535 1/20 0.33
MTOR P42345 2/20 0.32
PIK3C3 Q8NEB9 2/20 0.32
PDE4A P27815 1/20 0.32
ALDH1A1 P00352 2/20 0.32
SMN1; SMN2 Q16637 1/20 0.32
KDM4E B2RXH2 1/20 0.32
GAA P10253 2/20 0.32
HTT P42858 1/20 0.32
LTA4H P09960 3/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28025183 0.80 KCNMA1 (0.36) PIK3CDPIK3CANUDT1NPC1PDE4D
SCHEMBL27866878 0.74 GRIN2D (0.40) PIK3CDPIK3CAL3MBTL1ATRMTOR
SCHEMBL28025174 0.71 CHRNB2 (0.41) ATRMTORPIK3C3HTT
SCHEMBL30206003 0.70 AKR1C3 (0.46) ALDH1A1KDM4EGAA
SCHEMBL28024733 0.70 POLB (0.35) PIK3CDPIK3CANUDT1ALDH1A1SMN1; SMN2
SCHEMBL28025203 0.69 ATR (0.35) ATRPIK3C3ALDH1A1KDM4E
SCHEMBL137068 0.68 LMNA (0.47) PIK3C3ALDH1A1SMN1; SMN2KDM4E
SCHEMBL18988810 0.67 OPRL1 (0.36) PIK3CDPIK3CANUDT1PDE4DATR
SCHEMBL2096944 0.63 PIM1 (0.50) NPC1L3MBTL1ALDH1A1SMN1; SMN2KDM4E
SCHEMBL28821284 0.62 MTOR (0.36) PIK3CAATRMTORPIK3C3SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105143209-A Biaryl amide compounds as kinase inhibitors NOVARTIS AG 2015-12-09 CN disclosed