SCHEMBL28028683

SCHEMBL28028683

Cc1cc(C(=O)O)c(-c2cccc(Br)c2)c(C(=O)O)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TTR P02766 1/20 0.46
NPC1 O15118 3/20 0.46
RAB9A P51151 3/20 0.46
KMT2A Q03164 2/20 0.46
AURKA O14965 1/20 0.44
SORT1 Q99523 1/20 0.43
KDM4E B2RXH2 2/20 0.43
MYC P01106 2/20 0.43
SMN1; SMN2 Q16637 2/20 0.43
MEN1 O00255 1/20 0.43
GAA P10253 1/20 0.43
MAPT P10636 1/20 0.43
NPSR1 Q6W5P4 1/20 0.43
ALDH1A1 P00352 1/20 0.42
MAPK1 P28482 1/20 0.42
IKBKB O14920 1/20 0.42
AKR1C2 P52895 2/20 0.41
AKR1C1 Q04828 2/20 0.41
AKR1C3 P42330 1/20 0.41
FABP3 P05413 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27458636 0.82 TTR (0.59) TTRKMT2AKDM4EMEN1ALDH1A1
SCHEMBL27557477 0.81 RXFP1 (0.50) TTRNPC1KDM4EMYCMAPT
SCHEMBL27796625 0.80 TTR (0.46) TTRKMT2AKDM4EMEN1MAPT
SCHEMBL27631357 0.80 DHODH (0.58) TTRDHODHNR4A1
SCHEMBL28151298 0.78 SORT1 (0.43) NPC1RAB9AKMT2AAURKASORT1
SCHEMBL28201920 0.78 AKR1C2 (0.48) NPC1RAB9AKMT2AAURKASORT1
SCHEMBL27501023 0.78 GPR35 (0.56) KMT2AKDM4EALDH1A1AKR1C2AKR1C3
SCHEMBL27501021 0.76 PLAU (0.49) TTRTSHR
SCHEMBL17209586 0.74 ALDH1A1 (0.52) NPC1RAB9AKMT2AKDM4ESMN1; SMN2
SCHEMBL28565906 0.74 KMT2A (0.53) NPC1RAB9AKMT2AAURKASORT1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-104854108-A Pyrrolotriazinone derivatives as pi3k inhibitors ALMIRALL SA 2015-08-19 CN disclosed