SCHEMBL28036394

SCHEMBL28036394

Cc1ccc(-c2sc(C=O)c(-c3ccccc3)c2N)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.39
GRM6 O15303 5/20 0.37
KDM4E B2RXH2 4/20 0.36
MAPT P10636 4/20 0.36
LMNA P02545 2/20 0.36
MAPK1 P28482 2/20 0.36
NPSR1 Q6W5P4 2/20 0.36
XBP1 P17861 1/20 0.36
SMN1; SMN2 Q16637 1/20 0.36
ALDH1A1 P00352 6/20 0.36
MEN1 O00255 3/20 0.35
KMT2A Q03164 3/20 0.35
HPGD P15428 3/20 0.35
GRM5 P41594 1/20 0.34
RXFP1 Q9HBX9 1/20 0.33
AR P10275 1/20 0.33
RAB9A P51151 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2C9 P11712 1/20 0.33
CDK8 P49336 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27975859 0.91 ALDH1A1 (0.37) GRM6KDM4EMAPTLMNASMN1; SMN2
SCHEMBL28036416 0.87 PTGS2 (0.47) KDM4EMAPTLMNAMAPK1NPSR1
SCHEMBL27975579 0.85 TP53 (0.43) MAPTMAPK1MEN1KMT2ACYP1A2
SCHEMBL27975546 0.85 ALDH1A1 (0.40) GRM6KDM4EMAPTLMNAMAPK1
SCHEMBL27975865 0.83 TAAR1 (0.46) GRM6KDM4EMAPTLMNAALDH1A1
SCHEMBL28036417 0.82 ACHE (0.46) MAPTLMNAMAPK1NPSR1SMN1; SMN2
SCHEMBL28036395 0.81 ALDH1A1 (0.35) GRM6KDM4EMAPTLMNAMAPK1
SCHEMBL27975857 0.81 MAPT (0.52) MAPTLMNAMAPK1NPSR1SMN1; SMN2
SCHEMBL28036701 0.80 SIRT1 (0.40) KDM4EMAPTLMNANPSR1ALDH1A1
SCHEMBL27975539 0.77 ALDH1A1 (0.37) KDM4EMAPTLMNASMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103980248-B 3,5-bis-substituted-4-amino thiophene-2-formaldehyde compound and preparation method thereof ZHEJIANG UNIVERSITY (CN) 2015-11-18 CN disclosed