SCHEMBL28038733

SCHEMBL28038733

[N-]=[N+]=NCC(C(=O)C(CN=[N+]=[N-])c1cc(F)ccc1F)c1cc(F)ccc1F

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CES2 O00748 4/20 0.41
CES1 P23141 4/20 0.41
PSEN1 P49768 5/20 0.33
PSEN2 P49810 5/20 0.33
APH1B Q8WW43 5/20 0.33
NCSTN Q92542 5/20 0.33
APH1A Q96BI3 5/20 0.33
PSENEN Q9NZ42 5/20 0.33
PPARG P37231 1/20 0.32
PKM P14618 1/20 0.31
CA3 P07451 1/20 0.31
CA6 P23280 1/20 0.31
CA5A P35218 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
CA5B Q9Y2D0 1/20 0.31
RIPK1 Q13546 1/20 0.31
MAPT P10636 1/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
MDM2 Q00987 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27655951 0.78 HDAC3 (0.36)
SCHEMBL28038735 0.77 CES2 (0.35) CES2CES1PSEN1PSEN2APH1B
SCHEMBL27995445 0.70 CES2 (0.43) CES2CES1PSEN1PSEN2APH1B
SCHEMBL27719617 0.68 L3MBTL1 (0.41)
SCHEMBL17102138 0.68 CES2 (0.50) CES2CES1PPARGCA3CA6
SCHEMBL27723959 0.68 AURKA (0.33) SMN1; SMN2
SCHEMBL27953658 0.67 CES2 (0.46) CES2CES1PSEN1PSEN2APH1B
SCHEMBL28299886 0.67 TYR (0.44)
SCHEMBL21250530 0.66 CES2 (0.49) CES2CES1PSEN1PSEN2APH1B
SCHEMBL14270122 0.64 HTR2C (0.45) CES2CES1PSEN1PSEN2APH1B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105392772-B Preparation method of key intermediate of augustine 意大利合成制造有限公司 2017-09-15 CN disclosed
CN-105392772-A Preparation method of key intermediate of augustine FIS FABBRICA ITALIANA SINTETICI SPA 2016-03-09 CN disclosed