SCHEMBL27723959

SCHEMBL27723959

[N-]=[N+]=NCC(C(=O)C(CN=[N+]=[N-])c1ccccc1CN)c1ccccc1CN

nearest known ligand 0.33

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.33
RPS6KB1 P23443 1/20 0.33
GPR88 Q9GZN0 1/20 0.30
PNMT P11086 1/20 0.30
KDM4E B2RXH2 1/20 0.30
SMN1; SMN2 Q16637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27723961 0.77 PNMT (0.30) PNMT
SCHEMBL27656977 0.74 OPRM1 (0.36) PNMTKDM4ESMN1; SMN2
SCHEMBL27719617 0.74 L3MBTL1 (0.41) AURKARPS6KB1GPR88
SCHEMBL28264010 0.70 EPHX1 (0.39) PNMTKDM4ESMN1; SMN2
SCHEMBL28857685 0.68 CYP2C19 (0.47) AURKARPS6KB1GPR88SMN1; SMN2
SCHEMBL27473189 0.68 DPP4 (0.41) PNMTKDM4ESMN1; SMN2
SCHEMBL27723976 0.68 PPARG (0.40) KDM4ESMN1; SMN2
SCHEMBL28136810 0.67 KMT2A (0.38) PNMTKDM4ESMN1; SMN2
SCHEMBL28306686 0.67 CYP1A2 (0.54) KDM4ESMN1; SMN2
SCHEMBL28837383 0.67 ENPP2 (0.49) KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-102516192-A Antagonists of the vanilloid receptor subtype 1 (VR1) and uses thereof ABBOTT LAB 2012-06-27 CN disclosed
CN-101248052-A Vanilloid receptor subtype 1(VR1) antagonists and uses thereof ABBOTT LAB (US) 2008-08-20 CN disclosed