SCHEMBL28039573

SCHEMBL28039573

Clc1cc(Cl)c(-c2ccccc2)s1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 2/20 0.39
ESR1 P03372 1/20 0.38
ESR2 Q92731 1/20 0.38
CYP1A2 P05177 2/20 0.37
ALDH1A1 P00352 3/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
HPGD P15428 1/20 0.35
SMN1; SMN2 Q16637 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPT P10636 1/20 0.35
CYP2C19 P33261 1/20 0.35
ALOX5 P09917 1/20 0.34
LMNA P02545 1/20 0.33
TSHR P16473 1/20 0.33
CSNK2A1 P68400 1/20 0.33
HSP90AA1 P07900 1/20 0.33
NPC1 O15118 1/20 0.33
MAPK1 P28482 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4138504 0.80 HSD17B1 (0.44) CYP2A6ESR1ESR2CYP1A2ALDH1A1
SCHEMBL29290423 0.78 MAPK14 (0.38) CYP1A2MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL28087538 0.75 CYP2A6 (0.34) CYP2A6ESR1ESR2CYP1A2ALDH1A1
SCHEMBL13398620 0.74 DAO (0.55) ALDH1A1MEN1KMT2AHPGDSMN1; SMN2
SCHEMBL28087524 0.74 GRM6 (0.38) CYP2A6ESR1ALDH1A1MAPTALOX5
SCHEMBL5791411 0.71 PLA2G7 (0.44) ESR1ESR2CYP1A2ALDH1A1MEN1
SCHEMBL197250 0.68 CYP2A6 (0.61) CYP2A6ESR1CYP1A2ALDH1A1MEN1
SCHEMBL2932603 0.65 AHR (0.52) CYP2A6ESR2CYP1A2ALDH1A1MEN1
SCHEMBL544902 0.65 TDO2 (0.42) CYP2A6ESR1ALDH1A1MEN1KMT2A
SCHEMBL1895888 0.65 CASP3 (0.56) CYP2A6ESR1ESR2CYP1A2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-115151550-A Ectonucleotide pyrophosphatase/phosphodiesterase 1 (ENPP 1) modulators and uses thereof 桑福德·伯纳姆·普雷比医学发现研究所 2022-10-04 CN disclosed
CN-104011054-B As the thieno of potassium channel inhibitors and Furanopyrimidines class and pyridines 森申有限公司 2016-08-24 CN disclosed
CN-103492392-B Thieno [2,3-d ] pyrimidine derivatives and their use for the treatment of cardiac arrhythmias XENTION LTD. (GB) 2015-11-25 CN disclosed