Acridine

Acridine

SCHEMBL28040645

NC(=O)NSNC(=O)c1ccccc1.c1ccc2nc3ccccc3cc2c1

nearest known ligand 0.46

Full drug profile on Sugi Atlas →

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDR P35968 1/20 0.46
NPC1 O15118 4/20 0.46
RAB9A P51151 4/20 0.46
MAPT P10636 7/20 0.44
MEN1 O00255 4/20 0.44
KMT2A Q03164 4/20 0.44
SMN1; SMN2 Q16637 2/20 0.44
TP53 P04637 1/20 0.44
ALDH1A1 P00352 7/20 0.43
PLAU P00749 1/20 0.43
GLA P06280 1/20 0.43
HPGD P15428 1/20 0.43
ACHE P22303 1/20 0.43
IKBKB O14920 1/20 0.41
KDM4E B2RXH2 4/20 0.41
POLB P06746 4/20 0.41
GAA P10253 3/20 0.41
LMNA P02545 3/20 0.41
PABPC1 P11940 1/20 0.41
MAPK1 P28482 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27272343 0.84 ALDH1A1 (0.50) NPC1RAB9AMAPTKMT2AALDH1A1
Pyridine SCHEMBL28224545 0.79 JAK2 (0.47) MEN1KMT2ASMN1; SMN2TP53ALDH1A1
Acridine SCHEMBL4854060 0.76 ALDH1A1 (0.68) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL28343144 0.76 ALOX15 (0.58) NPC1RAB9AMAPTMEN1KMT2A
Benzophenone SCHEMBL30504146 0.72 ALDH1A1 (0.62) KDRNPC1RAB9AMAPTMEN1
Acridine SCHEMBL9644821 0.72 ALDH1A1 (0.62) KDRNPC1RAB9AMAPTMEN1
Benzil SCHEMBL9476443 0.72 ALDH1A1 (0.62) KDRNPC1RAB9AMAPTMEN1
Acridine SCHEMBL28228757 0.72 ALDH1A1 (0.68) NPC1RAB9AMAPTMEN1KMT2A
SCHEMBL2998471 0.72 KDM4E (0.55) KMT2ASMN1; SMN2TP53ALDH1A1KDM4E
SCHEMBL9131712 0.70 CYP1A2 (0.46) NPC1RAB9AMAPTMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105481769-B A kind of benzo (c) acridine derivatives and its preparation method and application 广西中医药大学 2018-07-10 CN disclosed
CN-105476992-B Application of the 2- methoxyl group -9- acridine benzamido thiocarbamides in acetylcholinesterase inhibitor is prepared 广西中医药大学 2018-07-06 CN disclosed
CN-105399670-B A kind of benzo (c) acridinium carboxamide base thiourea derivative and its preparation method and application 广西中医药大学 2018-04-17 CN disclosed
CN-105418608-B 7 benzos [b] [1,10] o-phenanthroline pyridinecarboxylic amido thiocarbamide and its production and use 广西中医药大学 2017-11-14 CN disclosed
CN-105481769-A Benzo(c)acridine derivative, and preparation method and use thereof UNIV GUANGXI CHINESE MEDICINE 2016-04-13 CN disclosed
CN-105418608-A 7-benzo[b]-[1,10]o-phenanthroline pyridine carboxamide thiourea as well as preparation method and application thereof UNIV GUANGXI CHINESE MEDICINE 2016-03-23 CN disclosed
CN-105399670-A Benzo[c]acridine amidothiourea derivative and preparation method and application thereof UNIV GUANGXI CHINESE MEDICINE 2016-03-16 CN disclosed