SCHEMBL28043008

SCHEMBL28043008

FC(F)(F)c1cccc(N2C=CC=NC2)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.45
HTR3E A5X5Y0 1/20 0.44
HTR3B O95264 1/20 0.44
HTR1D P28221 1/20 0.44
HTR2C P28335 1/20 0.44
HTR3A P46098 1/20 0.44
HTR3D Q70Z44 1/20 0.44
HTR3C Q8WXA8 1/20 0.44
SIGMAR1 Q99720 1/20 0.44
ALOX5 P09917 2/20 0.43
PTGS1 P23219 1/20 0.43
PTGS2 P35354 1/20 0.43
NOTUM Q6P988 4/20 0.43
MAPT P10636 3/20 0.43
THRB P10828 1/20 0.43
HTT P42858 1/20 0.41
EPHX2 P34913 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL32675963 0.85 NOTUM (0.36) NOTUM
SCHEMBL28249904 0.81 KIF11 (0.37) NOTUMMAPT
SCHEMBL28145993 0.80 KEAP1 (0.39) ALDH1A1HTR2CALOX5NOTUMMAPT
SCHEMBL27457816 0.76 MEN1 (0.41) ALDH1A1MEN1KMT2ALMNAKDM4E
SCHEMBL2362320 0.75 MAPT (0.35) ALDH1A1SIGMAR1MAPTHTTMEN1
SCHEMBL30642749 0.69 ALDH1A1 (0.41) ALDH1A1MAPTHTTMEN1KMT2A
SCHEMBL28918666 0.69 DHFR (0.30)
SCHEMBL28261507 0.68 MAPK1 (0.33) ALDH1A1NOTUMMAPTHTTMEN1
SCHEMBL28254340 0.68
SCHEMBL28178897 0.68 CYP2A6 (0.40) MAPTHTT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105121442-A PI3K and/or mTOR inhibitor prodrug XUANZHU PHARMA CO LTD 2015-12-02 CN disclosed