SCHEMBL28145993

SCHEMBL28145993

Fc1cccc(N2C=CC=NC2)c1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KEAP1 Q14145 1/20 0.39
FAAH O00519 1/20 0.39
MGLL Q99685 1/20 0.39
NOTUM Q6P988 1/20 0.38
MAPT P10636 2/20 0.36
ALDH1A1 P00352 1/20 0.36
POLB P06746 1/20 0.36
GAA P10253 1/20 0.36
MEN1 O00255 1/20 0.35
KMT2A Q03164 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
ALOX5 P09917 1/20 0.35
BPTF Q12830 1/20 0.34
RXRA P19793 1/20 0.33
GRIN1 Q05586 1/20 0.33
GRIN2B Q13224 1/20 0.33
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33
HTR2B P41595 1/20 0.33
PI4KA P42356 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28254340 0.82
SCHEMBL22588493 0.81 HTR1A (0.33) FAAHMGLLALDH1A1
SCHEMBL27457816 0.80 MEN1 (0.41) ALDH1A1POLBMEN1KMT2ALMNA
SCHEMBL28043008 0.80 ALDH1A1 (0.45) NOTUMMAPTALDH1A1GAAMEN1
SCHEMBL28261507 0.79 MAPK1 (0.33) MGLLNOTUMMAPTALDH1A1MEN1
SCHEMBL2362320 0.78 MAPT (0.35) MAPTALDH1A1GAAMEN1KMT2A
SCHEMBL32675963 0.76 NOTUM (0.36) KEAP1NOTUMNFE2L2
SCHEMBL28171948 0.72 FAAH (0.41) KEAP1FAAHMGLLNOTUMMAPT
SCHEMBL28918666 0.72 DHFR (0.30)
SCHEMBL28178897 0.71 CYP2A6 (0.40) MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-103889962-B Substituted n-(3-(pyrimidin-4-yl)phenyl)acrylamide analogs as tyrosine receptor kinase BTK inhibitors 犹他大学研究基金会 2017-05-03 CN disclosed