SCHEMBL28044047

SCHEMBL28044047

COc1cc(N(CCC[C](C)C)C(C)=O)ccc1N

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.40
CYP3A4 P08684 2/20 0.40
TSHR P16473 2/20 0.38
HSD17B10 Q99714 1/20 0.38
TDP1 Q9NUW8 1/20 0.38
KMT2A Q03164 1/20 0.37
MAPK1 P28482 1/20 0.36
ATM Q13315 1/20 0.36
MTNR1A P48039 1/20 0.36
MTNR1B P49286 1/20 0.36
HTT P42858 1/20 0.36
MAPK3 P27361 1/20 0.36
TSPO P30536 1/20 0.36
KCNH2 Q12809 1/20 0.36
MET P08581 2/20 0.35
ACHE P22303 2/20 0.35
GPX4 P36969 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28824480 0.84 ALDH1A1 (0.41) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL15938081 0.83 MTNR1A (0.40) ALDH1A1CYP3A4TSHRMTNR1AMTNR1B
SCHEMBL15938784 0.82 SMN1; SMN2 (0.48) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL17102727 0.81 ACHE (0.36) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL15938676 0.80 MTNR1A (0.42) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL28043962 0.78 AR (0.40) MAPK3ACHE
SCHEMBL17102736 0.78 ACHE (0.37) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL28824481 0.75 MAPK3 (0.49) MTNR1AMTNR1BMAPK3
SCHEMBL28824484 0.75 MET (0.35) ALDH1A1CYP3A4TSHRHSD17B10TDP1
SCHEMBL15938665 0.74 ALDH1A1 (0.33) ALDH1A1CYP3A4TSHRHSD17B10TDP1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105188371-A Erk inhibitors and uses thereof CELGENE AVILOMICS RES INC 2015-12-23 CN disclosed