SCHEMBL28045762

SCHEMBL28045762

O=C(Cc1ccccc1)N[C@@H](CC(C(=O)O)C(=O)OCc1ccccc1)C(=O)O

nearest known ligand 0.48

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CNR2 P34972 4/20 0.48
ALDH1A1 P00352 1/20 0.47
MAPK1 P28482 1/20 0.47
L3MBTL1 Q9Y468 1/20 0.47
CASP1 P29466 1/20 0.46
ITGB3 P05106 1/20 0.46
ITGA2B P08514 1/20 0.46
CTSB P07858 2/20 0.44
ACE P12821 1/20 0.44
CTSL P07711 1/20 0.44
CTSS P25774 1/20 0.44
PSMB8 P28062 2/20 0.44
PSMB5 P28074 2/20 0.44
MBTPS1 Q14703 1/20 0.44
GPR34 Q9UPC5 1/20 0.44
NAALAD2 Q9Y3Q0 1/20 0.43
POLB P06746 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9831107 0.87 CNR2 (0.57) CNR2ALDH1A1ITGB3ITGA2BCTSB
SCHEMBL9831110 0.87 CNR2 (0.57) CNR2ALDH1A1ITGB3ITGA2BCTSB
SCHEMBL10660589 0.81 ALDH1A1 (0.51) CNR2ALDH1A1MAPK1L3MBTL1CASP1
SCHEMBL13819263 0.81 ACE (0.63) CNR2ALDH1A1MAPK1L3MBTL1ITGB3
SCHEMBL18775036 0.81 CTSK (0.57) ALDH1A1CTSBCTSLCTSSPSMB8
SCHEMBL18791070 0.81 CTSK (0.57) ALDH1A1CTSBCTSLCTSSPSMB8
SCHEMBL24339778 0.80 FOLH1 (0.48) CTSBNAALAD2
SCHEMBL7347418 0.80 CASP1 (0.60) CNR2ALDH1A1MAPK1L3MBTL1CASP1
SCHEMBL28045721 0.78 FOLH1 (0.63) CNR2ITGB3ITGA2BCTSBCTSL
SCHEMBL28045720 0.78 FOLH1 (0.63) CNR2ITGB3ITGA2BCTSBCTSL

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105175418-B Pentacyclic indole quinolizine for inhibiting autophagy of cells, synthesis, antitumor activity and application thereof 首都医科大学 2020-01-14 CN disclosed
CN-105175418-A Pentacyclic indole quinolizine inhibiting cell autophagy, synthesis, antitumor activity and application thereof UNIV CAPITAL MEDICAL SCIENCES 2015-12-23 CN disclosed