SCHEMBL28046258

SCHEMBL28046258

Nc1cncc(Cc2cc(F)cc(F)c2)n1

nearest known ligand 0.40

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NOS1 P29475 10/20 0.40
NOS3 P29474 6/20 0.40
NOS2 P35228 8/20 0.36
CDK2 P24941 1/20 0.35
IDO1 P14902 2/20 0.34
BACE1 P56817 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28000659 0.83 NPC1 (0.47) NOS1NOS3NOS2IDO1
SCHEMBL9391584 0.74 GRM4 (0.43) NOS1NOS3NOS2CDK2
SCHEMBL28810940 0.73 IDO1 (0.35) NOS1NOS3IDO1BACE1
SCHEMBL28040110 0.68 ALDH1A1 (0.51) IDO1
SCHEMBL14814345 0.66 CLK1 (0.37)
SCHEMBL14642748 0.66
SCHEMBL11400820 0.66
SCHEMBL12466519 0.66 MBOAT4 (0.37) BACE1
SCHEMBL5251885 0.66 IDO1 (0.50) IDO1
SCHEMBL21384229 0.66 GABRP (0.44) NOS3NOS2IDO1BACE1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105324380-A Pyrrolo[2,3-b]pyridine cdk9 kinase inhibitors ABBVIE INC 2016-02-10 CN disclosed