SCHEMBL28046429

SCHEMBL28046429

CC(C)(C)C(=O)ON1CCC(c2cccc(Br)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DRD2 P14416 2/20 0.42
DRD1 P21728 1/20 0.42
DRD4 P21917 1/20 0.42
DRD5 P21918 1/20 0.42
DRD3 P35462 1/20 0.42
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
RIPK1 Q13546 2/20 0.39
PDE5A O76074 1/20 0.38
HDAC4 P56524 1/20 0.38
HRH3 Q9Y5N1 1/20 0.38
ALDH1A1 P00352 2/20 0.36
TP53 P04637 1/20 0.36
NAMPT P43490 1/20 0.36
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
RECQL P46063 1/20 0.36
KDM4E B2RXH2 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28258134 0.88 TSHR (0.40) DRD2DRD1DRD4DRD5DRD3
SCHEMBL27682015 0.84 RIPK1 (0.39) DRD2RIPK1NAMPTKCNQ2QDPR
SCHEMBL27629058 0.83 NAMPT (0.41) RIPK1ALDH1A1NAMPTPOLBQDPR
SCHEMBL27488566 0.83 RIPK1 (0.51) DRD2RIPK1HRH3ALDH1A1NAMPT
SCHEMBL28017548 0.83 DRD2 (0.54) DRD2TSHRALDH1A1LMNAKDM4E
SCHEMBL27635041 0.81 DRD3 (0.49) DRD2DRD3TSHRNPSR1
SCHEMBL30014833 0.81 NAMPT (0.53) NAMPTKDM4E
SCHEMBL1427529 0.81 NAMPT (0.53) NAMPTKDM4E
SCHEMBL28059420 0.80 LMNA (0.46) ALDH1A1LMNARECQL
SCHEMBL27724744 0.80 HDAC1 (0.38) RIPK1HDAC4NAMPTQDPR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105209457-A Pyrrolidine derivatives, pharmaceutical compositions containing them, and their use in therapy ABBVIE DEUTSCHLAND 2015-12-30 CN disclosed