SCHEMBL27682015

SCHEMBL27682015

CC(C)(C)C(=O)ON1CCC(c2cccc(N)c2)CC1

nearest known ligand 0.42

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
RIPK1 Q13546 3/20 0.39
DRD2 P14416 2/20 0.36
CHRNB2 P17787 1/20 0.36
CHRNA4 P43681 1/20 0.36
PARP10 Q53GL7 1/20 0.36
NAMPT P43490 1/20 0.36
KCNQ2 O43526 1/20 0.35
QDPR P09417 1/20 0.35
SLC18A3 Q16572 2/20 0.35
BCL9 O00512 1/20 0.35
CTNNB1 P35222 1/20 0.35
KMO O15229 1/20 0.35
DDB1 Q16531 1/20 0.35
CRBN Q96SW2 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL27872124 0.87 DRD3 (0.41) DRD2BCL9CTNNB1
SCHEMBL28046429 0.84 DRD2 (0.42) RIPK1DRD2NAMPTKCNQ2QDPR
SCHEMBL27318172 0.83 SLC18A3 (0.44) RIPK1NAMPTQDPRSLC18A3DDB1
SCHEMBL27488566 0.83 RIPK1 (0.51) RIPK1DRD2NAMPTSLC18A3
SCHEMBL28017548 0.83 DRD2 (0.54) DRD2BCL9CTNNB1
SCHEMBL28294631 0.83 HDAC1 (0.40) RIPK1NAMPTQDPR
SCHEMBL27635041 0.81 DRD3 (0.49) DRD2
SCHEMBL30376009 0.81 GPR119 (0.54) NAMPTDDB1CRBN
SCHEMBL28024448 0.81 OPRL1 (0.36) CRBN
SCHEMBL835855 0.81 GPR119 (0.54) NAMPTDDB1CRBN

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 9 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105849096-B Piperidine derivatives having multimodal activity against pain 埃斯蒂文制药股份有限公司 2019-11-29 CN disclosed
CN-104736533-B Vegfr3 inhibitor 癌症治疗合作研究中心有限公司 2016-12-07 CN disclosed
CN-105849096-A Piperidine derivatives having multimodal activity against pain 埃斯蒂文博士实验室股份有限公司 2016-08-10 CN disclosed
CN-105384695-A Pyrimidine derivative, preparation method therefor and application thereof in medicine SICHUAN HAISCO PHARMACEUTICAL CO LTD 2016-03-09 CN disclosed
CN-103534241-B Fak inhibitor Cancer Therapeutics CRC Pty Ltd. (AU) 2015-11-25 CN disclosed
CN-104837835-A VEGFR3 inhibitors CANCER THERAPEUTICS CRC PTY LTD 2015-08-12 CN disclosed
CN-103534241-A Fak inhibitor CANCER THERAPEUTICS CRC PTY LTD 2014-01-22 CN disclosed
CN-102459258-A Preparation and use of 1,2, 4-triazolo [1,5a ] pyridine derivatives CEPHALON INC 2012-05-16 CN disclosed
CN-101052629-A Aryl-amino substituted pyrrolopyrimidine multi-kinase inhibiting compounds OSI PHARM INC (US) 2007-10-10 CN disclosed