SCHEMBL28258134

SCHEMBL28258134

CC(C)(C)C(=O)ON1CC(c2cccc(Br)c2)C1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 1/20 0.40
NPSR1 Q6W5P4 1/20 0.40
DRD2 P14416 1/20 0.40
DRD1 P21728 1/20 0.40
DRD4 P21917 1/20 0.40
DRD5 P21918 1/20 0.40
DRD3 P35462 1/20 0.40
PDE5A O76074 1/20 0.39
HDAC4 P56524 1/20 0.39
SLC6A4 P31645 1/20 0.37
SLC6A3 Q01959 1/20 0.37
LMNA P02545 1/20 0.36
POLB P06746 1/20 0.36
RECQL P46063 1/20 0.36
KDM1A O60341 3/20 0.36
RCOR1 Q9UKL0 1/20 0.35
HTR2A P28223 1/20 0.35
HTR2C P28335 1/20 0.35
HTR2B P41595 1/20 0.35
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28046429 0.88 DRD2 (0.42) TSHRNPSR1DRD2DRD1DRD4
SCHEMBL28024239 0.83 BRD4 (0.42) NPSR1PDE5ASLC6A4SLC6A3LMNA
SCHEMBL19385185 0.78 RORC (0.49) DRD2DRD1DRD4DRD5DRD3
SCHEMBL27979570 0.74 SLC18A3 (0.33) TSHRLMNAALDH1A1RIPK1
SCHEMBL28790708 0.74 PDE5A (0.36) TSHRNPSR1PDE5ALMNAPOLB
SCHEMBL27958057 0.74 HTT (0.43) TSHRSLC6A4SLC6A3POLBKDM1A
SCHEMBL27979665 0.74 ACMSD (0.52) POLBRECQLALDH1A1ALOX5
SCHEMBL28822639 0.73 ALDH1A1 (0.36) TSHRLMNAALDH1A1RIPK1
SCHEMBL28103918 0.73 USP30 (0.41) TSHRDRD2PDE5ALMNARECQL
SCHEMBL21381960 0.73 DRD2 (0.48) TSHRNPSR1DRD2DRD1DRD4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-108884068-A 1- cyano-pyrolidin derivative as DUB inhibitor 特殊治疗有限公司 2018-11-23 CN disclosed