SCHEMBL28051139

SCHEMBL28051139

CCn1c2ccc([N+](=O)[O-])cc2c2cc(S(=O)(=O)Nc3cc(OC)c(OC)c(OC)c3)ccc21

nearest known ligand 0.51

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 6/20 0.51
KMT2A Q03164 6/20 0.51
MAPT P10636 5/20 0.51
LMNA P02545 4/20 0.51
ALDH1A1 P00352 7/20 0.49
HTT P42858 3/20 0.49
SMN1; SMN2 Q16637 3/20 0.49
TP53 P04637 1/20 0.45
THRB P10828 1/20 0.45
POLB P06746 3/20 0.44
HPGD P15428 2/20 0.44
L3MBTL1 Q9Y468 1/20 0.44
KDM4E B2RXH2 1/20 0.43
MAPK1 P28482 2/20 0.42
PKM P14618 1/20 0.42
TSHR P16473 1/20 0.42
HTR6 P50406 1/20 0.42
PTGS2 P35354 1/20 0.41
KDR P35968 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL23148487 0.85 MAPT (0.61) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL28051135 0.85 HTT (0.52) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL28252795 0.83 HTT (0.50) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL6343830 0.80 MEN1 (0.67) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL6342356 0.78 HTT (0.46) MEN1KMT2ALMNAALDH1A1HTT
SCHEMBL6342525 0.76 ALDH1A1 (0.68) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL148001 0.75 MAPT (0.85) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL29539965 0.75 MAPT (0.85) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL28051137 0.73 HTT (0.61) MEN1KMT2AMAPTLMNAALDH1A1
SCHEMBL6340645 0.72 TUBB4A (0.56) MAPTLMNAALDH1A1HTTSMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 6 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN claimed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN claimed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN claimed
CN-105287388-B High dispersive carbazole sulfonamide derivative and preparation method thereof 山西普德药业有限公司 2019-09-17 CN disclosed
CN-105418487-A Carbazole sulfonamide derivative eutectic and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-03-23 CN disclosed
CN-105287388-A High-dispersion carbazole sulfonamide derivatives and preparation method thereof SHANXI PUDE PHARMACEUTICS CO LTD 2016-02-03 CN disclosed